SCHEMBL26109002

SCHEMBL26109002

O=C(O)c1ccc(-c2cc3c(=O)nc[nH]c3[nH]2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CSF1R P07333 2/20 0.39
GRIK1 P39086 1/20 0.39
GRIK2 Q13002 1/20 0.39
GRIK3 Q13003 1/20 0.39
GCGR P47871 1/20 0.39
MAPK14 Q16539 1/20 0.39
MAPKAPK2 P49137 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
CAMKK2 Q96RR4 2/20 0.37
AXL P30530 2/20 0.37
SGK1 O00141 1/20 0.37
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26521358 0.84 KDM4E (0.46) KDM4EALDH1A1CSF1RMAPKAPK2CAMKK2
SCHEMBL4372018 0.70 HTR7 (0.47) KDM4EALDH1A1CSNK2A1
SCHEMBL8870966 0.70 CSNK2A1 (0.49) KDM4EALDH1A1CSNK2A1
SCHEMBL4071289 0.67 EGFR (0.58) EGFRCSF1R
SCHEMBL13627444 0.65 PARP1 (0.36)
SCHEMBL6638123 0.64 CYP3A4 (0.60) KDM4EALDH1A1
SCHEMBL22283252 0.63 PDE3B (0.46) ALDH1A1
SCHEMBL700288 0.62 MAPT (0.62) EGFRKDM4EALDH1A1GRIK1GRIK2
SCHEMBL3072721 0.61 NOTUM (0.66) EGFRKDM4EALDH1A1GRIK1GRIK2
Terephthalic Acid SCHEMBL9577834 0.60 TSHR (0.80) EGFRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023183652-A1 DUAL CXCR4-BTK INHIBITORS X4 PHARMACEUTICALS, INC. (US) 2023-09-28 WO disclosed