SCHEMBL261232

SCHEMBL261232

CC(C)(C(=O)O)c1ccc(NC(N)=O)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 7/20 0.64
PEPD P12955 1/20 0.52
MAPT P10636 2/20 0.52
GAA P10253 1/20 0.52
GFER P55789 1/20 0.52
ALDH1A1 P00352 3/20 0.50
NPC1 O15118 1/20 0.50
CYP26A1 O43174 1/20 0.47
CYP26B1 Q9NR63 1/20 0.47
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL262075 0.86 KIF11 (0.51) KIF11MAPTGAAALDH1A1CYP26A1
SCHEMBL10683046 0.83 SMN1; SMN2 (0.56) MAPTGAAALDH1A1NPC1CYP26A1
SCHEMBL2191366 0.82 KIF11 (0.89) KIF11PEPDMAPTALDH1A1NPC1
SCHEMBL3497043 0.79 MAPT (0.52) MAPTALDH1A1CYP26A1CYP26B1HDAC3
SCHEMBL5425660 0.78 KIF11 (1.00) KIF11PEPDMAPTNPC1HDAC3
SCHEMBL5062623 0.77 PEPD (0.80) KIF11PEPDMAPTGAAGFER
SCHEMBL23343691 0.76 KIF11 (0.62) KIF11PEPDMAPTGAAGFER
SCHEMBL167549 0.75 KIF11 (0.89) KIF11PEPDMAPTALDH1A1NPC1
SCHEMBL2875784 0.75 NPC1 (0.61) KIF11PEPDMAPTGAAGFER
SCHEMBL31510753 0.75 KMT2A (0.50) KIF11MAPTALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8133911-B2 (R)-4-(heteroaryl) phenylethyl derivatives and pharmaceutical compositions containing them DOMPE S.P.A (IT) 2012-03-13 US disclosed
EP-2201006-B1 (R)-4-(HETEROARYL) PHENYLETHYL DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DOMPE SPA (IT) 2011-03-09 EP disclosed