SCHEMBL262075

SCHEMBL262075

CC(C)(C(=O)O)c1ccc(NC(N)=S)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.51
ALDH1A1 P00352 4/20 0.50
TP53 P04637 1/20 0.50
TYR P14679 1/20 0.50
TSHR P16473 1/20 0.50
TAS2R38 P59533 1/20 0.50
HSD17B10 Q99714 1/20 0.50
MAPT P10636 2/20 0.47
KMT2A Q03164 2/20 0.47
GAA P10253 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
ALOX12 P18054 2/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
HPGD P15428 1/20 0.46
CYP2C19 P33261 1/20 0.46
CYP26A1 O43174 1/20 0.45
CYP26B1 Q9NR63 1/20 0.45
HDAC3 O15379 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL261232 0.86 KIF11 (0.64) KIF11ALDH1A1MAPTKMT2AGAA
SCHEMBL10683046 0.80 SMN1; SMN2 (0.56) ALDH1A1TSHRHSD17B10MAPTKMT2A
SCHEMBL4348957 0.80 KIF11 (0.59) KIF11ALDH1A1TP53TYRTSHR
SCHEMBL3497043 0.77 MAPT (0.52) ALDH1A1TSHRMAPTKMT2ACYP2D6
SCHEMBL12071196 0.76 CYP17A1 (0.51) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL12070405 0.75 ALDH1A1 (0.64) KIF11ALDH1A1TP53TYRTSHR
SCHEMBL725810 0.74 ALDH1A1 (0.75) KIF11ALDH1A1TP53TYRTSHR
SCHEMBL23987221 0.74 KIF11 (0.53) KIF11ALDH1A1TP53TYRTSHR
SCHEMBL5458028 0.74 SMN1; SMN2 (0.61) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL27477483 0.73 KIF11 (0.42) KIF11ALDH1A1TP53TYRTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346841-B1 2-ARYL-PROPIONIC ACIDS AND DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DOMPÉ S P A (IT) 2015-01-14 EP claimed
US-8133911-B2 (R)-4-(heteroaryl) phenylethyl derivatives and pharmaceutical compositions containing them DOMPE S.P.A (IT) 2012-03-13 US disclosed
EP-2201006-B1 (R)-4-(HETEROARYL) PHENYLETHYL DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DOMPE SPA (IT) 2011-03-09 EP disclosed