SCHEMBL26133607

SCHEMBL26133607

COc1c(Br)cnc([N+](=O)[O-])c1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.43
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35
GRIN3A Q8TCU5 1/20 0.35
TPMT P51580 2/20 0.35
GPR35 Q9HC97 1/20 0.33
ERN1 O75460 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
AMY1A P0DUB6 1/20 0.32
HTT P42858 2/20 0.32
POLB P06746 1/20 0.32
PKM P14618 1/20 0.32
ALDH1A1 P00352 2/20 0.32
LMNA P02545 1/20 0.32
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30413667 1.00 MAPT (0.43) MAPTGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL31347289 0.78 MAPT (0.46) MAPTGPR35SMN1; SMN2HTTALDH1A1
SCHEMBL3285272 0.78 MAPT (0.49) MAPTGPR35ERN1ALDH1A1LMNA
SCHEMBL25246827 0.73 GRIN2D (0.43) MAPTGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL31683208 0.72 GRIN2D (0.42) MAPTGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL27190094 0.72 CTSB (0.40) MAPTTPMTGPR35ERN1SMN1; SMN2
SCHEMBL16475125 0.71 KDM4E (0.37) MAPTGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL30325942 0.70 PDXK (0.35) TPMTPOLB
SCHEMBL21383944 0.70 KMT2A (0.38) MAPTGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL29947327 0.70 KMT2A (0.38) MAPTGRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023066825-A1 FUSED BICYCLIC HETEROARYL COMPOUNDS USEFUL AS NLRP3 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2023-04-27 WO disclosed