SCHEMBL2616331

SCHEMBL2616331

Cc1noc(CNC(=O)C2CN(C)c3ccccc3O2)n1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
RAB9A P51151 2/20 0.43
HPGD P15428 6/20 0.41
HTT P42858 1/20 0.41
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
KDM1A O60341 1/20 0.40
MAOA P21397 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
NPC1 O15118 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4830461 0.79 HPGD (0.60) ALDH1A1RAB9AHPGDHTTTSHR
SCHEMBL11544729 0.74 KMT2A (0.48) ALDH1A1RAB9AHPGDHTTTSHR
SCHEMBL29586755 0.74 HDAC4 (0.45) ALDH1A1RAB9AHPGDHTTSMN1; SMN2
SCHEMBL24496705 0.74 HDAC4 (0.45) ALDH1A1RAB9AHPGDHTTSMN1; SMN2
SCHEMBL2685855 0.69 SIRT1 (0.58)
SCHEMBL31566197 0.69 SIRT1 (0.58)
SCHEMBL925260 0.69 SIRT1 (0.48) ALDH1A1RAB9AHPGDHTTSMN1; SMN2
SCHEMBL1689630 0.69 KMT2A (0.55) ALDH1A1HPGDSMN1; SMN2
SCHEMBL7820037 0.68 POLB (0.53) ALDH1A1HTTTSHRSMN1; SMN2POLB
SCHEMBL18581461 0.67 HPGD (0.47) ALDH1A1RAB9AHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8202858-B2 Vasopressin V1a antagonists VANTIA LIMITED (GB) 2012-06-19 US disclosed
US-8202858-B2 Vasopressin V1a antagonists VANTIA LIMITED (GB) 2012-06-19 US disclosed
US-20120101082-A1 VASOPRESSIN V1A ANTAGONISTS BATT ANDRZEJ ROMAN (GB) 2012-04-26 US disclosed
US-20120101082-A1 VASOPRESSIN V1A ANTAGONISTS BATT ANDRZEJ ROMAN (GB) 2012-04-26 US disclosed
US-20090029965-A1 Vasopressin V1a Antagonists FERRING B.V. (NL) 2009-01-29 US disclosed
US-20090029965-A1 Vasopressin V1a Antagonists FERRING B.V. (NL) 2009-01-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120101082-A1 VASOPRESSIN V1A ANTAGONISTS AVPR1A, AVPR2, AVPR1B ALDH1A1 902/4885RAB9A 668/4885HPGD 286/4885
US-20090029965-A1 Vasopressin V1a Antagonists AVPR1A, AVPR2, AVPR1B ALDH1A1 902/4885RAB9A 668/4885HPGD 286/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.