SCHEMBL26317142

SCHEMBL26317142

CNC(=O)c1c(O)cccc1NC=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.43
CA1 P00915 4/20 0.43
CA2 P00918 4/20 0.43
CA7 P43166 4/20 0.43
CA9 Q16790 4/20 0.43
CA14 Q9ULX7 4/20 0.43
THRB P10828 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
TAS1R2 Q8TE23 1/20 0.40
KDM5A P29375 2/20 0.39
HTT P42858 4/20 0.36
GAA P10253 3/20 0.36
PLK1 P53350 1/20 0.36
PLK3 Q9H4B4 1/20 0.36
MAPT P10636 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20880608 0.82 GAA (0.46) HTTGAAPLK1PLK3KMT2A
SCHEMBL6501339 0.80 CA12 (0.58) CA12CA1CA2CA7CA9
SCHEMBL29954290 0.76 ERN1 (0.50) CA12CA1CA2CA7CA9
SCHEMBL28031204 0.73 ESR2 (0.47) CA12CA1CA2CA7CA9
SCHEMBL3567350 0.72 ERN1 (0.48) CA1CA2KDM5AHTTGAA
SCHEMBL29876843 0.72 GAA (0.50) CA12CA2CA14KDM5AHTT
SCHEMBL1939410 0.72 GAA (0.50) CA12CA2CA14KDM5AHTT
SCHEMBL13354976 0.70 CA12 (0.47) CA12CA1CA2CA7CA9
SCHEMBL11207914 0.69 TSHR (0.44) CA1CA2KDM5AHTTGAA
SCHEMBL8989665 0.69 G6PD (0.42) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3960735-B1 QUINAZOLINE DERIVATIVES USED TO TREAT HIV GILEAD SCIENCES INC (US) 2023-09-13 EP disclosed