SCHEMBL2635686

SCHEMBL2635686

[CH2]CCNCc1ccc(-c2ccc(CCCCCC)cc2)c(-c2cocn2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 16/20 0.43
S1PR1 P21453 9/20 0.36
S1PR2 O95136 7/20 0.36
LPAR2 Q9HBW0 3/20 0.36
S1PR4 O95977 4/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HSD17B10 Q99714 1/20 0.33
S1PR5 Q9H228 1/20 0.33
SPNS2 Q8IVW8 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL35951 0.86 S1PR3 (0.63) S1PR3S1PR1S1PR2LPAR2S1PR4
SCHEMBL36123 0.69 S1PR3 (0.66) S1PR3S1PR1S1PR2LPAR2S1PR4
SCHEMBL36337 0.68 S1PR3 (0.87) S1PR3S1PR1S1PR2LPAR2S1PR4
SCHEMBL13279803 0.68 S1PR1 (0.43) S1PR3S1PR1S1PR2LPAR2S1PR4
SCHEMBL35933 0.67 S1PR3 (0.67) S1PR3S1PR1S1PR2LPAR2S1PR4
SCHEMBL27939769 0.67 HTR5A (0.41) S1PR3S1PR1S1PR2LPAR2S1PR4
SCHEMBL27939768 0.67 HTR5A (0.41) S1PR3S1PR1S1PR2LPAR2S1PR4
SCHEMBL19217017 0.59 S1PR1 (0.73) S1PR3S1PR1S1PR2LPAR2S1PR4
SCHEMBL6736726 0.59 HSD17B10 (0.55) KDM4EMEN1USP2ALDH1A1GAA
SCHEMBL10462640 0.59 MAPT (0.55) KDM4EMEN1USP2ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2569322-A1 AROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHONATE (S1P) RECEPTOR ACTIVITY Allergan, Inc. (US) 2013-03-20 EP disclosed
WO-2011143332-A1 AROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHONATE (S1P) RECEPTOR ACTIVITY ALLERGAN, INC. (US) 2011-11-17 WO disclosed