SCHEMBL2638515

SCHEMBL2638515

Cc1cc(S(N)(=O)=O)ccc1NC(=O)Cc1ccc(C)c(Oc2cc(Cl)ccc2Br)c1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA1 P00915 15/20 0.58
CA2 P00918 15/20 0.58
CA12 O43570 12/20 0.58
CA9 Q16790 12/20 0.58
CTSD P07339 3/20 0.48
CA5A P35218 3/20 0.47
CA7 P43166 3/20 0.47
CA5B Q9Y2D0 3/20 0.47
EPAS1 Q99814 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2639161 0.89 CA2 (0.59) CA1CA2CA12CA9CA5A
SCHEMBL2638680 0.82 CA1 (0.52) CA1CA2CA12CA9CTSD
SCHEMBL2638641 0.82 MEN1 (0.53) CA1CA2CA12CA9
SCHEMBL2638936 0.80 CA1 (0.48) CA1CA2CA12CA9CTSD
SCHEMBL2638624 0.79 CA1 (0.61) CA1CA2CA12CA9CA5A
SCHEMBL2639110 0.79 CA12 (0.42) CA1CA2CA12CA9
SCHEMBL2639656 0.79 CA1 (0.58) CA1CA2CA12CA9CA5A
SCHEMBL2638562 0.78 CTSD (0.48) CA1CA2CA12CA9CTSD
SCHEMBL2639453 0.78 CA1 (0.61) CA1CA2CA12CA9CA5A
SCHEMBL4602432 0.77 CA12 (0.42) CA1CA2CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4810529-B2 2011-11-09 JP claimed
EP-1742908-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP claimed
EP-1742908-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-01-17 EP claimed
WO-2005102989-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2005-11-03 WO claimed
EP-1742908-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP disclosed