SCHEMBL2641322

SCHEMBL2641322

COc1cc(OC)cc(OCCOc2nccnc2N2CCNCC2)c1.COc1ccccc1OCCOc1nccnc1N1CCNCC1.Fc1ccc(F)c(OCCOc2nccnc2N2CCNCC2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.40
HTR6 P50406 3/20 0.38
ADRB1 P08588 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CYP2C19 P33261 2/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
HTR3A P46098 1/20 0.36
HTR3D Q70Z44 1/20 0.36
HTR3C Q8WXA8 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4312678 0.87 HTR2C (0.41) HTR2CHTR6SLC6A2SLC6A4HTR1A
SCHEMBL6046287 0.86 CCNT1 (0.42) HTR2CHTR6ADRB1CYP2C19USP2
SCHEMBL4312809 0.84 CYP2C19 (0.49) HTR2CHTR6ADRB1CYP2C19USP2
SCHEMBL4309052 0.82 ADRB1 (0.50) HTR6ADRB1CYP2C19USP2CYP1A2
SCHEMBL7474730 0.81 CYP2C19 (0.48) HTR2CHTR6ADRB1CYP2C19USP2
SCHEMBL4320202 0.80 HTR2C (0.50) HTR2CHTR6CYP2C19ALDH1A1CYP1A2
SCHEMBL2641702 0.79 HTR2C (0.42) HTR2CHTR6ADRB1CYP2C19USP2
SCHEMBL4319475 0.79 HTR2C (0.42) HTR2CHTR6ALDH1A1SLC6A2SLC6A4
SCHEMBL4322355 0.79 HTR2C (0.50) HTR2CHTR6SLC6A2HTR1A
SCHEMBL4315672 0.78 ADRB1 (0.52) HTR2CHTR6ADRB1CYP2C19USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4831903-B2 2011-12-07 JP claimed
EP-1178973-A2 NOVEL COMPOUNDS, THEIR USE AND PREPARATION Pharmacia AB (SE) 2002-02-13 EP claimed
WO-2000076984-A2 NOVEL COMPOUNDS, THEIR USE AND PREPARATION BIOVITRUM AB (SE) 2000-12-21 WO claimed