SCHEMBL2641702

SCHEMBL2641702

COc1cccc(OCCOc2nccnc2N2CCNCC2)c1.Fc1ccccc1OCCOc1nccnc1N1CCNCC1.N#Cc1cccc(OCCOc2nccnc2N2CCNCC2)c1.c1ccc(OCCOc2nccnc2N2CCNCC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.42
CYP1A2 P05177 4/20 0.38
HTR6 P50406 3/20 0.38
CYP3A4 P08684 3/20 0.38
TP53 P04637 2/20 0.38
CYP2D6 P10635 2/20 0.38
TSHR P16473 2/20 0.38
ICMT O60725 2/20 0.38
ADRB1 P08588 1/20 0.37
LMNA P02545 1/20 0.37
BCL2A1 Q16548 1/20 0.36
USP2 O75604 2/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MAPK1 P28482 1/20 0.36
CASP1 P29466 1/20 0.36
HIF1A Q16665 1/20 0.36
TBXAS1 P24557 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4317771 0.85 HTR2C (0.52) HTR2CCYP1A2HTR6CYP3A4TP53
SCHEMBL4315672 0.83 ADRB1 (0.52) HTR2CCYP1A2HTR6CYP3A4TP53
SCHEMBL4320202 0.81 HTR2C (0.50) HTR2CCYP1A2HTR6CYP3A4CYP2D6
SCHEMBL7476206 0.80 ADRB1 (0.51) HTR2CCYP1A2HTR6CYP3A4TP53
SCHEMBL2641322 0.79 HTR2C (0.40) HTR2CCYP1A2HTR6CYP3A4ADRB1
SCHEMBL7601597 0.78 ADRB1 (0.47) HTR2CCYP1A2HTR6CYP3A4TP53
SCHEMBL2640084 0.77 CHRNB2 (0.49) HTR2CCYP1A2HTR6CYP3A4TP53
SCHEMBL4308039 0.77 TSHR (0.48) HTR2CHTR6TSHRHSD17B10
SCHEMBL4316292 0.76 SLC6A2 (0.47) HTR2CHTR6ADRB1LMNACYP2C19
SCHEMBL4316373 0.75 HTR2C (0.55) HTR2CCYP1A2CYP3A4LMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4831903-B2 2011-12-07 JP claimed
EP-1178973-A2 NOVEL COMPOUNDS, THEIR USE AND PREPARATION Pharmacia AB (SE) 2002-02-13 EP claimed
WO-2000076984-A2 NOVEL COMPOUNDS, THEIR USE AND PREPARATION BIOVITRUM AB (SE) 2000-12-21 WO claimed