SCHEMBL26414747

SCHEMBL26414747

O=C(NC1CCCCC1)c1c[nH]c2ccccc12

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.76
NPC1 O15118 6/20 0.76
ALDH1A1 P00352 5/20 0.58
KMT2A Q03164 3/20 0.58
BACE1 P56817 1/20 0.57
KDM4E B2RXH2 2/20 0.56
LMNA P02545 2/20 0.56
TDP1 Q9NUW8 1/20 0.56
HPGD P15428 1/20 0.56
HTT P42858 1/20 0.56
HDAC1 Q13547 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
SMN1; SMN2 Q16637 3/20 0.55
MEN1 O00255 2/20 0.55
MAPK1 P28482 1/20 0.55
HTR3E A5X5Y0 1/20 0.55
HTR3B O95264 1/20 0.55
HTR3A P46098 1/20 0.55
HTR3D Q70Z44 1/20 0.55
HTR3C Q8WXA8 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20590676 0.86 RAB9A (0.59) RAB9ANPC1ALDH1A1KMT2AKDM4E
SCHEMBL21489827 0.86 RAB9A (0.59) RAB9ANPC1ALDH1A1HPGDHTT
SCHEMBL19710504 0.86 RAB9A (0.59) RAB9ANPC1ALDH1A1HPGDHTT
SCHEMBL8314705 0.82 RAB9A (0.55) RAB9ANPC1ALDH1A1KMT2ABACE1
SCHEMBL21489781 0.82 SMYD3 (0.70) RAB9ANPC1HPGDHTTHDAC1
SCHEMBL19710071 0.82 SMYD3 (0.70) RAB9ANPC1HPGDHTTHDAC1
SCHEMBL25224750 0.82 ALDH1A1 (0.59) RAB9ANPC1ALDH1A1KMT2AKDM4E
SCHEMBL5265256 0.81 RAB9A (0.57) RAB9ANPC1ALDH1A1KMT2ABACE1
SCHEMBL29176340 0.81 ALDH1A1 (0.54) RAB9ANPC1ALDH1A1KMT2ABACE1
SCHEMBL9235867 0.81 RAB9A (0.56) RAB9ANPC1ALDH1A1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023192901-A9 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-12-14 WO disclosed
WO-2023192901-A1 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-10-05 WO disclosed