SCHEMBL26415237

SCHEMBL26415237

CC(C)Cc1nc2cnccc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.51
KDM4E B2RXH2 1/20 0.51
GSK3B P49841 1/20 0.46
AAK1 Q2M2I8 3/20 0.43
KDM4C Q9H3R0 2/20 0.40
MAPK1 P28482 3/20 0.40
ALPL P05186 2/20 0.40
DDAH1 O94760 1/20 0.39
CYP3A4 P08684 3/20 0.36
CYP2D6 P10635 3/20 0.36
CYP2C9 P11712 3/20 0.36
CYP2C19 P33261 3/20 0.36
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
TP53 P04637 2/20 0.36
ALOX12 P18054 1/20 0.36
TSHR P16473 1/20 0.36
KRAS P01116 1/20 0.36
CYP1A2 P05177 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12088725 0.87 KDM4E (0.55) MAPTKDM4EGSK3BAAK1MAPK1
SCHEMBL10206036 0.81 DDAH1 (0.59) KDM4CDDAH1KRASHTT
SCHEMBL19001265 0.80 PKM (0.42) KDM4EAAK1KDM4CMAPK1ALPL
SCHEMBL9851482 0.78 KDM4C (0.63) KDM4EAAK1KDM4CDDAH1KMT2A
SCHEMBL4072911 0.77 CACNA1H (0.44) KDM4CDDAH1KRAS
SCHEMBL7578581 0.77 KDM4C (0.40) KDM4EKDM4CDDAH1KRASSMN1; SMN2
SCHEMBL31875233 0.77 CACNA1H (0.44) KDM4CDDAH1KRAS
SCHEMBL5806722 0.77 TDP1 (0.49) KDM4CDDAH1KRASNPSR1TDP1
SCHEMBL4113303 0.77 DDAH1 (0.65) MAPTKDM4EMAPK1ALPLDDAH1
SCHEMBL11955037 0.77 KDM4C (0.40) AAK1KDM4CDDAH1CYP2C9KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3675858-B1 IMIDAZO[1,5-A]PYRAZINE COMPOUNDS AND COMPOSITIONS FOR IRE1 INHIBITION OPTIKIRA LLC (US) 2023-04-26 EP disclosed