Tolfenpyrad

Tolfenpyrad

SCHEMBL26416

CCc1nn(C)c(C(=O)NCc2ccc(Oc3ccc(C)cc3)cc2)c1Cl

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.57
SMN1; SMN2 Q16637 4/20 0.57
LMNA P02545 4/20 0.57
KMT2A Q03164 2/20 0.57
GALR3 O60755 1/20 0.57
NR2F2 P24468 1/20 0.57
MAPK14 Q16539 2/20 0.50
MMP13 P45452 2/20 0.49
CYP3A4 P08684 2/20 0.49
MMP2 P08253 1/20 0.49
STAT3 P40763 1/20 0.49
HTT P42858 1/20 0.49
L3MBTL1 Q9Y468 2/20 0.46
CHRNA7 P36544 1/20 0.45
NPC1 O15118 4/20 0.43
ALPL P05186 1/20 0.43
ALPI P09923 1/20 0.43
ALPG P10696 1/20 0.43
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20384620 0.87 SMN1; SMN2 (0.41) RAB9ASMN1; SMN2LMNAKMT2AGALR3
Tolfenpyrad SCHEMBL16541149 0.87 KMT2A (0.46) RAB9ASMN1; SMN2LMNAKMT2AGALR3
Tolfenpyrad SCHEMBL27825694 0.87 MAPK14 (0.46) RAB9ASMN1; SMN2LMNAKMT2AGALR3
SCHEMBL8077552 0.85 LMNA (0.54) RAB9ASMN1; SMN2LMNAKMT2AGALR3
SCHEMBL28925367 0.84 LMNA (0.53) RAB9ASMN1; SMN2LMNAKMT2AGALR3
SCHEMBL15220664 0.84 LMNA (0.60) RAB9ASMN1; SMN2LMNAKMT2AGALR3
SCHEMBL30150564 0.82 RAB9A (0.46) RAB9ASMN1; SMN2LMNAKMT2AGALR3
SCHEMBL30150619 0.81 LMNA (0.46) RAB9ASMN1; SMN2LMNAKMT2AGALR3
Tolfenpyrad SCHEMBL28139546 0.81 MAPK14 (0.40) RAB9ASMN1; SMN2LMNAKMT2AGALR3
SCHEMBL10061335 0.81 LMNA (0.57) RAB9ASMN1; SMN2LMNAKMT2AGALR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 20127 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4734762-A1 BAIT COMPOSITIONS FMC Corporation (US) 2026-05-06 EP claimed
WO-2026088131-A1 STABLE SYNERGISTIC PESTICIDAL COMPOSITION COMPRISING TOLFENPYRAD, ETHION, AND PYRIPROXYFEN RANI SANGEETA (IN) 2026-04-30 WO claimed
EP-4719059-A1 INCREASED PALATABILITY OF INSECTICIDAL INSECT BAITS Bio Logic Crop Science, S.L. (ES) 2026-04-08 EP claimed
US-20260083130-A1 NOVEL SULFONATE BENZAMIDE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS FMC CORP (US) 2026-03-26 US claimed
US-20260083129-A1 PYRAZOLE AMIDE INSECTICIDES FMC CORP (US) 2026-03-26 US claimed
EP-4710766-A1 MIXTURES OF AMBRUTICIN WITH AT LEAST ONE FURTHER PESTICIDE BASF SE (DE) 2026-03-18 EP claimed
EP-4709166-A1 NOVEL INSECTICIDAL MIXTURES FOR CONTROLLING AND PROTECTING CROPS ADAMA MAKHTESHIM LTD. (IL) 2026-03-18 EP claimed
US-12568969-B2 Pyridine compounds for controlling invertebrate pests FMC CORPORATION (US) 2026-03-10 US claimed
CN-121577800-A Non-targeted screening multi-pesticide residue detection method based on high-resolution mass spectrum 常州市食品药品纤维质量监督检验中心(常州市粮油质量监督检测站、常州纤维检验所) 2026-02-27 CN claimed
CN-121586714-A Connected bicyclic compounds for control and combating invertebrate pests FMC公司 2026-02-27 CN claimed
WO-2005080327-A1 INSECTICIDAL AND NEMATICIDAL DIFLUOROALKENE DERIVATIVES E.I. DUPONT DE NEMOURS AND COMPANY (US) 2005-09-01 WO claimed
EP-1328154-B1 PESTICIDAL COMPOSITION ISHIHARA SANGYO KAISHA (JP) 2005-07-27 EP claimed
WO-2005053407-A1 PESTICIDALLY ACTIVE COMBINATIONS SYNGENTA PARTICIPATIONS AG (CH) 2005-06-16 WO claimed
WO-2004082382-A1 SYNERGISTIC HERBICIDAL COMPOSITION COMPRISING A HERBICIDALLY ACTIVE COMPOUND IN COMBINATION WITH AN INSECTICIDE SYNGENTA PARTICIPATIONS AG (CH) 2004-09-30 WO claimed
WO-2004067528-A1 CYANO ANTHRANILAMIDE INSECTICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 2004-08-12 WO claimed
US-20040078843-A1 Method for controlling harmful organisms in the culture of useful plants BAYER CROPSCIENCE GMBH (DE) 2004-04-22 US claimed
EP-1367900-A2 METHOD FOR CONTROLLING HARMFUL ORGANISMS IN THE CULTURE OF USEFUL PLANTS Bayer CropScience GmbH (DE) 2003-12-10 EP claimed
US-20030198659-A1 Fibrous pest control CORNELL RESEARCH FOUNDATION, INC. 2003-10-23 US claimed
WO-2002062144-A2 METHOD FOR CONTROLLING HARMFUL ORGANISMS IN THE CULTURE OF USEFUL PLANTS BAYER CROPSCIENCE GMBH (DE) 2002-08-15 WO claimed
WO-2001056358-A2 ENHANCED PROPERTIED PESTICIDES ROHM AND HAAS COMPANY (US) 2001-08-09 WO claimed