SCHEMBL264163

SCHEMBL264163

[2H]/C(C(=O)OC)=C(\[2H])C([2H])([2H])[C@@]([2H])(CO[Si](c1ccccc1)(c1ccccc1)C(C)(C)C)NC(=O)OCc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSL P07711 10/20 0.40
CTSS P25774 9/20 0.40
CTSB P07858 6/20 0.40
CTSK P43235 7/20 0.38
ATM Q13315 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ALOX15 P16050 1/20 0.37
KYNU Q16719 1/20 0.37
SYK P43405 1/20 0.37
MBOAT4 Q96T53 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2793720 0.93 CTSS (0.41) CTSLCTSSCTSBCTSKATM
SCHEMBL263479 0.83 CTSL (0.41) CTSLCTSSCTSBCTSKATM
SCHEMBL2794568 0.83 CTSS (0.43) CTSLCTSSCTSBCTSKATM
SCHEMBL15924777 0.77 KYNU (0.53) CTSLCTSSCTSBCTSKATM
SCHEMBL15924778 0.77 KYNU (0.53) CTSLCTSSCTSBCTSKATM
SCHEMBL5724195 0.77 SYK (0.52) CTSLCTSSCTSBCTSKATM
SCHEMBL23455702 0.76 PPARA (0.51) CTSLCTSSCTSBCTSKATM
SCHEMBL10045788 0.76 PPARA (0.51) CTSLCTSSCTSBCTSKATM
SCHEMBL5724014 0.76 ATM (0.50) CTSLCTSSCTSBCTSKATM
SCHEMBL262927 0.76 SYK (0.47) CTSLCTSSCTSBCTSKATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8133908-B2 Heteroaryl derivatives of N-{[(1S,4S,6S)-3-(2-pyridinylcarbonyl)-3-azabicyclo[4.1.0]hept-4-yl]methyl}-2-amine GLAXO GROUP LIMITED (GB) 2012-03-13 US disclosed
EP-2370427-A1 N-{[(IR,4S,6R-3-(2-PYRIDINYLCARBONYL)-3-AZABICYCLO [4.1.0]HEPT-4-YL]METHYL}-2-HETEROARYLAMINE DERIVATIVES AND USES THEREOF Glaxo Group Limited (GB) 2011-10-05 EP disclosed