SCHEMBL26418792

SCHEMBL26418792

CNS(=O)(=O)c1cc(F)ccc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSTO1 P78417 1/20 0.51
MCL1 Q07820 5/20 0.46
MGAM O43451 1/20 0.44
VCAM1 P19320 1/20 0.42
NR3C1 P04150 1/20 0.41
PGR P06401 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA3 P07451 1/20 0.41
CA4 P22748 1/20 0.41
CA6 P23280 1/20 0.41
CA5A P35218 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA13 Q8N1Q1 1/20 0.41
CA14 Q9ULX7 1/20 0.41
CA5B Q9Y2D0 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12932911 0.82 ALDH1A1 (0.47) MCL1MGAMNR3C1PGRHPGD
SCHEMBL10153817 0.81 SMN1; SMN2 (0.48) NR3C1LMNACCR2
SCHEMBL2372705 0.81 MCL1 (0.62) GSTO1MCL1CA12CA1CA2
SCHEMBL11512510 0.79 MCL1 (0.61) GSTO1MCL1CA12CA1CA2
SCHEMBL2525525 0.79 LMNA (0.65) MCL1LMNA
SCHEMBL13855836 0.79 GSTO1 (0.53) GSTO1MCL1VCAM1CA12CA1
SCHEMBL11512517 0.79 MCL1 (0.61) GSTO1MCL1CA12CA1CA2
SCHEMBL9322506 0.78 GSTO1 (0.51) GSTO1MCL1VCAM1CA12CA1
SCHEMBL9322517 0.78 KMT2A (0.56) GSTO1MCL1VCAM1CA12CA1
SCHEMBL375209 0.78 ALDH1A1 (0.42) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3675858-B1 IMIDAZO[1,5-A]PYRAZINE COMPOUNDS AND COMPOSITIONS FOR IRE1 INHIBITION OPTIKIRA LLC (US) 2023-04-26 EP disclosed