SCHEMBL2641968

SCHEMBL2641968

CC(=O)Nc1cccc(-c2cccc(-n3cnc4cc(C(F)(F)F)ccc43)c2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.62
RAB9A P51151 3/20 0.62
SMN1; SMN2 Q16637 2/20 0.55
AURKA O14965 2/20 0.54
AURKB Q96GD4 2/20 0.54
KDR P35968 1/20 0.54
FGFR1 P11362 6/20 0.51
ALDH1A1 P00352 3/20 0.51
HPGD P15428 2/20 0.51
LMNA P02545 2/20 0.51
FYN P06241 1/20 0.48
ATM Q13315 1/20 0.47
GABRA1 P14867 1/20 0.46
GABRG2 P18507 1/20 0.46
GABRB3 P28472 1/20 0.46
GABRA5 P31644 1/20 0.46
GABRA3 P34903 1/20 0.46
ADRA2B P18089 1/20 0.46
SYK P43405 1/20 0.46
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2340937 0.82 NPC1 (0.59) NPC1RAB9ASMN1; SMN2FGFR1HPGD
SCHEMBL1761988 0.80 GABRA1 (0.56) NPC1RAB9ASMN1; SMN2AURKAAURKB
SCHEMBL2653352 0.79 NPC1 (0.53) NPC1RAB9ASMN1; SMN2AURKAAURKB
SCHEMBL2641981 0.78 FGFR1 (0.56) SMN1; SMN2AURKAAURKBKDRFGFR1
SCHEMBL7989436 0.78 NPC1 (1.00) NPC1RAB9ASMN1; SMN2FGFR1ALDH1A1
Hydrochloric Acid SCHEMBL2641992 0.77 FGFR1 (0.54) SMN1; SMN2AURKAAURKBKDRFGFR1
Diethylamine SCHEMBL2642037 0.77 KDR (0.48) NPC1RAB9ASMN1; SMN2KDRFGFR1
Hydrochloric Acid SCHEMBL7976246 0.77 NPC1 (0.97) NPC1RAB9ASMN1; SMN2FGFR1ALDH1A1
SCHEMBL4503339 0.76 NPC1 (0.70) NPC1RAB9ASMN1; SMN2FGFR1ALDH1A1
SCHEMBL2642007 0.76 HPGD (0.49) NPC1RAB9ASMN1; SMN2AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0563001-B1 Imidazole compounds, their preparation and use NEUROSEARCH AS (DK) 1996-02-28 EP disclosed
US-5360809-A Imidazole compounds and their use as calcium channel blockers NEUROSEARCH A/S (DK) 1994-11-01 US disclosed
EP-0563001-A1 Imidazole compounds, their preparation and use NEUROSEARCH A/S (DK) 1993-09-29 EP disclosed