SCHEMBL2643655

SCHEMBL2643655

c1ccc(CCc2c[nH]nn2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.50
NOS1 P29475 1/20 0.41
BACE1 P56817 1/20 0.40
MAOB P27338 4/20 0.39
TAAR1 Q96RJ0 2/20 0.39
MAOA P21397 3/20 0.39
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38
CASP1 P29466 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NISCH Q9Y2I1 1/20 0.38
ATM Q13315 1/20 0.38
DAO P14920 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
TDP1 Q9NUW8 2/20 0.37
CYP2A6 P11509 1/20 0.37
HTR2A P28223 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27892139 0.89 HTR2A (0.42) KCNH2NOS1MAOBMAOADAO
SCHEMBL29869051 0.87 HTR2A (0.41) KCNH2NOS1MAOBMAOADAO
SCHEMBL28221103 0.87 HTR2A (0.41) KCNH2NOS1MAOBMAOADAO
SCHEMBL29272 0.82 ALDH1A1 (0.46) MAOBTAAR1ALDH1A1HPGDRAB9A
Benzene SCHEMBL27499662 0.82 ALDH1A1 (0.46) MAOBTAAR1ALDH1A1HPGDRAB9A
SCHEMBL11066734 0.80 TSHR (0.45) TAAR1ALDH1A1NPC1RAB9ATDP1
SCHEMBL9508013 0.80 ALDH1A1 (0.44) MAOBTAAR1ALDH1A1HPGDRAB9A
Nitrous Acid SCHEMBL28299073 0.79 HDAC8 (0.38) NOS1MAOBMAOADAOHTR2A
SCHEMBL10469971 0.78 HTR1A (0.62)
SCHEMBL28026394 0.77 TSHR (0.56) NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 88 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797093-B1 NOVEL 3-METHYL-7-BUTINYL-XANTHINES, PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM INT (DE) 2012-05-30 EP claimed
EP-0842158-A1 MICROBICIDAL 2-PHENYLETHYL-MERCAPTO-TRIAZOLES BAYER AG (DE) 1998-05-20 EP claimed
WO-1997005119-A1 MICROBICIDAL 2-PHENYLETHYL-MERCAPTO-TRIAZOLES BAYER AKTIENGESELLSCHAFT (DE) 1997-02-13 WO claimed
US-4921870-A Fungicidal novel substituted phenethyl-triazolyl derivatives BAYER AKTIENGESELLSCHAFT (DE) 1990-05-01 US claimed
US-4771065-A Fungicidal novel substituted phenethyl-triazolyl derivatives BAYER AKTIENGESELLSCHAFT (DE) 1988-09-13 US claimed
EP-0119572-B1 SUBSTITUTED PHENETHYL-TRIAZOLYL DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS FUNGICIDES BAYER AG (DE) 1988-08-10 EP claimed
EP-0000017-B1 1-(2-PHENYLETHYL)-TRIAZOLIUM SALTS, THEIR PREPARATION AND THEIR USE AS FUNGICIDES BAYER AG (DE) 1981-09-30 EP claimed
EP-0000018-B1 METAL SALT COMPLEXES OF 1-PHENYL-2-TRIAZOLYL-ETHANE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES BAYER AG (DE) 1981-01-07 EP claimed
CN-113754601-B Synthesis method of N2-beta-sulfanyl triazole derivative 周口师范学院 2023-04-11 CN disclosed
CN-113754601-A Synthesis method of N2-beta-sulfanyl triazole derivative 周口师范学院 2021-12-07 CN disclosed
EP-2167491-A1 5-HETEROARYL SUBSTITUTED INDAZOLES AS KINASE INHIBITORS Abbott Laboratories (US) 2010-03-31 EP disclosed
US-7495002-B2 3-methyl-7-butinyl-xanthines, the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-02-24 US disclosed
WO-2008154241-A1 5-HETEROARYL SUBSTITUTED INDAZOLES AS KINASE INHIBITORS ABBOTT LABORATORIES (US) 2008-12-18 WO disclosed
EP-1121361-B1 PYRAZOLO-TRIAZINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME (GB) 2007-08-29 EP disclosed
EP-0063099-B1 PROCESS FOR THE PREPARATION OF PHENYLETHYL TRIAZOLES CIBA-GEIGY AG (CH) 1985-11-27 EP disclosed
EP-0119572-A2 Substituted phenethyl-triazolyl derivatives, process for their preparation and their use as fungicides BAYER AG (DE) 1984-09-26 EP disclosed
US-4366152-A Combatting fungi with metal salt complexes of 1-phenyl-2-(1,2,4-triazol-1-yl)-ethanes BAYER AKTIENGESELLSCHAFT (DE) 1982-12-28 US disclosed
EP-0063099-A2 Process for the preparation of phenylethyl triazoles CIBA-GEIGY AG (CH) 1982-10-20 EP disclosed
EP-0000018-B1 METAL SALT COMPLEXES OF 1-PHENYL-2-TRIAZOLYL-ETHANE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES BAYER AG (DE) 1981-01-07 EP disclosed
EP-0000018-A1 Metal salt complexes of 1-phenyl-2-triazolyl-ethane derivatives, their preparation and their use as fungicides BAYER AG (DE) 1978-12-20 EP disclosed