SCHEMBL26466925

SCHEMBL26466925

COc1cc(NC(=O)CN2C[C@@H]3C[C@H]2CN3CC(=O)NC(C)(C)C)cc(F)c1F

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 5/20 0.46
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 1/20 0.38
ANO1 Q5XXA6 1/20 0.38
WNT3A P56704 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
LTA4H P09960 1/20 0.36
GFER P55789 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KMT2A Q03164 1/20 0.35
CXCR6 O00574 1/20 0.35
IMPDH2 P12268 1/20 0.35
IMPDH1 P20839 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26466996 0.89 CACNA1H (0.41) CACNA1HALDH1A1KDM4EANO1LTA4H
SCHEMBL26466777 0.88 ALDH1A1 (0.45) CACNA1HALDH1A1KDM4EANO1WNT3A
SCHEMBL26466921 0.85 CACNA1H (0.41) CACNA1HTSHRHTTLTA4HKMT2A
SCHEMBL26466922 0.84 CACNA1H (0.41) CACNA1HALDH1A1KDM4EWNT3ATSHR
SCHEMBL26466617 0.82 CACNA1H (0.67) CACNA1HALDH1A1KDM4ELTA4HLMNA
SCHEMBL26466913 0.82 L3MBTL1 (0.48) CACNA1HALDH1A1KDM4EHTTLTA4H
SCHEMBL26466596 0.79 CACNA1H (0.40) CACNA1HALDH1A1KDM4EANO1HTT
SCHEMBL26466613 0.78 CACNA1H (0.52) CACNA1HALDH1A1ANO1LTA4HMAPT
SCHEMBL26466398 0.78 CACNA1H (0.49) CACNA1HALDH1A1ANO1LTA4H
SCHEMBL26466390 0.78 CACNA1H (0.49) CACNA1HALDH1A1ANO1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023192669-A1 T-TYPE CALCIUM CHANNEL MODULATORS COMPRISING A PIPERAZINE OR 1,4-DIAZEPANE CORE AND METHODS OF USE THEREOF PRAXIS PRECISION MEDICINES, INC. (US) 2023-10-05 WO disclosed