SCHEMBL2646800

SCHEMBL2646800

O=Cc1ccc(C(=O)NCCC(=O)O)cc1.O=Cc1ccc(C(=O)NCCC(=O)O)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.58
CA2 P00918 3/20 0.58
MAPK1 P28482 1/20 0.57
ALDH1A1 P00352 2/20 0.50
EPHX2 P34913 1/20 0.50
NR1H4 Q96RI1 1/20 0.50
SIRT5 Q9NXA8 2/20 0.48
NME4 O00746 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
CHRM1 P11229 1/20 0.48
ADORA2A P29274 1/20 0.48
AVPR2 P30518 1/20 0.48
AGTR1 P30556 1/20 0.48
SLC6A4 P31645 1/20 0.48
AVPR1A P37288 1/20 0.48
HTR3A P46098 1/20 0.48
GCDH Q92947 1/20 0.48
SLC29A1 Q99808 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
HRH3 Q9Y5N1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2646881 1.00 CA1 (0.58) CA1CA2MAPK1ALDH1A1EPHX2
SCHEMBL16688444 0.89 MAPK1 (0.76) CA1CA2MAPK1ALDH1A1EPHX2
SCHEMBL9717434 0.87 MAPK1 (0.71) CA1CA2MAPK1ALDH1A1SIRT5
SCHEMBL12989840 0.85 EPHX2 (0.52) CA1CA2MAPK1ALDH1A1EPHX2
SCHEMBL2646805 0.83 PRSS1 (0.66) CA1CA2MAPK1ALDH1A1EPHX2
SCHEMBL1664008 0.82 POLB (0.53) CA1CA2MAPK1ALDH1A1EPHX2
SCHEMBL1765747 0.82 ALDH1A1 (0.53) ALDH1A1EPHX2NR1H4PRSS1CTSG
SCHEMBL13760114 0.82 CA1 (0.54) CA1CA2MAPK1EPHX2NR1H4
SCHEMBL22042366 0.81 MAPK1 (0.51) MAPK1ALDH1A1EPHX2NR1H4LMNA
SCHEMBL2654472 0.81 UNG (0.56) CA1CA2MAPK1PRSS1CTSG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005058845-A2 NOVEL GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 2005-06-30 WO disclosed
EP-1463715-A1 NOVEL GLUCAGON ANTAGONISTS NOVO NORDISK A/S (DK) 2004-10-06 EP disclosed
WO-2003048109-A1 NOVEL GLUCAGON ANTAGONISTS NOVO NORDISK A/S (DK) 2003-06-12 WO disclosed