SCHEMBL26468205

SCHEMBL26468205

CON(C)C(=O)c1ncc(F)cc1Br

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 1/20 0.36
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
MLYCD O95822 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
AGBL2 Q5U5Z8 1/20 0.33
KEAP1 Q14145 1/20 0.32
PKM P14618 1/20 0.32
GPBAR1 Q8TDU6 1/20 0.32
CLK1 P49759 1/20 0.31
DYRK1A Q13627 1/20 0.31
DYRK1B Q9Y463 1/20 0.31
PIK3CA P42336 1/20 0.31
MTOR P42345 1/20 0.31
PDK2 Q15119 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30296581 1.00 TRPM8 (0.36) TRPM8MEN1KMT2AMLYCDTDP1
SCHEMBL568769 0.84 PDK2 (0.40) TRPM8MLYCDAGBL2GPBAR1CLK1
SCHEMBL14484964 0.83 KDM4E (0.36) MEN1KMT2AMLYCDTDP1CLK1
SCHEMBL24424181 0.79 MLYCD (0.38) TRPM8MEN1KMT2AMLYCDGPBAR1
SCHEMBL30133796 0.79 MLYCD (0.38) TRPM8MEN1KMT2AMLYCDGPBAR1
SCHEMBL2943288 0.79 MLYCD (0.36) TRPM8MEN1KMT2AMLYCDTDP1
SCHEMBL16632434 0.78 NPSR1 (0.41) AGBL2KEAP1PKM
SCHEMBL30960730 0.78 NPSR1 (0.41) AGBL2KEAP1PKM
SCHEMBL29560615 0.75 AGBL2 (0.39) AGBL2KEAP1PKM
SCHEMBL22866557 0.75 AGBL2 (0.39) AGBL2KEAP1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916754-A Heteroaromatic macrocyclic ether chemotherapeutic agents 纽威伦特公司 2023-04-04 CN disclosed