SCHEMBL2648414

SCHEMBL2648414

CC(=O)c1ccc(Nc2cccc(-c3ccccn3)c2)c(N)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.49
GAA P10253 2/20 0.49
ALDH1A1 P00352 2/20 0.49
MAPT P10636 2/20 0.49
KDM4E B2RXH2 1/20 0.49
THRB P10828 1/20 0.49
HPGD P15428 1/20 0.49
HSD17B10 Q99714 1/20 0.49
AKR1C3 P42330 3/20 0.48
AKR1C2 P52895 3/20 0.48
ATR Q13535 1/20 0.47
SYK P43405 1/20 0.47
NPC1 O15118 3/20 0.46
GFER P55789 1/20 0.46
AKR1B10 O60218 1/20 0.46
AKR1B1 P15121 1/20 0.46
AKR1C4 P17516 1/20 0.46
AKR1C1 Q04828 1/20 0.46
PRKCI P41743 1/20 0.46
ERBB2 P04626 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2647819 0.83 HCAR3 (0.53) CNR1ALDH1A1MAPTHPGDAKR1C3
SCHEMBL2650071 0.82 GAA (0.49) GAAALDH1A1MAPTKDM4ETHRB
SCHEMBL2655100 0.81 GAA (0.46) GAAALDH1A1MAPTKDM4ETHRB
SCHEMBL2643439 0.81 NPC1 (0.53) CNR1GAAALDH1A1MAPTKDM4E
SCHEMBL30937997 0.80 MAP4K4 (0.55) CNR1ALDH1A1KDM4ESYKNPC1
SCHEMBL17742695 0.80 MAP4K4 (0.55) CNR1ALDH1A1KDM4ESYKNPC1
SCHEMBL2645152 0.80 RET (0.45) CNR1GAAALDH1A1MAPTKDM4E
SCHEMBL2647667 0.79 GAA (0.48) CNR1GAAALDH1A1MAPTKDM4E
SCHEMBL7989959 0.79 GAA (0.77) GAAALDH1A1MAPTKDM4ETHRB
SCHEMBL2652430 0.77 AKR1C3 (0.45) GAAALDH1A1MAPTKDM4ETHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821682-B1 BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS MODULATORS OF THE GABA-A RECEPTOR COMPLEX NEUROSEARCH AS (DK) 2000-07-19 EP disclosed
US-5922725-A Benzimidazole compounds and their use as modulators of the GABAA receptor complex NEUROSEARCH A/S (DK) 1999-07-13 US disclosed
EP-0821682-A1 BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS MODULATORS OF THE GABA A? RECEPTOR COMPLEX NEUROSEARCH A/S (DK) 1998-02-04 EP disclosed
WO-1996033191-A1 BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS MODULATORS OF THE GABAA RECEPTOR COMPLEX NEUROSEARCH A/S (DK) 1996-10-24 WO disclosed