Phenazopyridine

Phenazopyridine

SCHEMBL26499

Cl.Nc1ccc(N=Nc2ccccc2)c(N)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9A

The experimentally established mechanism targets of Phenazopyridine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 1.00
MEN1 O00255 8/20 1.00
KMT2A Q03164 8/20 1.00
MAPK1 P28482 6/20 1.00
TDP1 Q9NUW8 5/20 1.00
CYP3A4 P08684 3/20 1.00
SMN1; SMN2 Q16637 3/20 1.00
HBB P68871 2/20 1.00
KDM4E B2RXH2 2/20 1.00
TSHR P16473 2/20 1.00
ALOX15 P16050 2/20 1.00
SARM1 Q6SZW1 1/20 1.00
HSD17B10 Q99714 1/20 1.00
LMNA P02545 3/20 0.96
CYP1A2 P05177 2/20 0.96
HIF1A Q16665 2/20 0.96
USP2 O75604 1/20 0.96
CHRM1 P11229 1/20 0.96
CYP2C9 P11712 1/20 0.96
DRD2 P14416 1/20 0.96

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenazopyridine SCHEMBL14687482 1.00 MAPT (1.00) MAPTMEN1KMT2AMAPK1TDP1
Phenazopyridine SCHEMBL29392321 1.00 MAPT (1.00) MAPTMEN1KMT2AMAPK1TDP1
Phenazopyridine SCHEMBL28796595 1.00 MAPT (1.00) MAPTMEN1KMT2AMAPK1TDP1
Phenazopyridine SCHEMBL215655 1.00 MAPT (1.00) MAPTMEN1KMT2AMAPK1TDP1
Phenazopyridine SCHEMBL19357 1.00 MAPT (1.00) MAPTMEN1KMT2AMAPK1TDP1
Phenazopyridine SCHEMBL301672 0.98 MAPT (0.96) MAPTMEN1KMT2AMAPK1TDP1
Phenazopyridine SCHEMBL5973732 0.98 MAPT (0.96) MAPTMEN1KMT2AMAPK1TDP1
Phenazopyridine SCHEMBL302506 0.98 MAPT (0.96) MAPTMEN1KMT2AMAPK1TDP1
Phenazopyridine SCHEMBL6661856 0.98 MAPT (0.96) MAPTMEN1KMT2AMAPK1TDP1
Phenazopyridine SCHEMBL9151827 0.98 MAPT (0.96) MAPTMEN1KMT2AMAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2295 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4709723-A1 ISOXAZOLIDINES AS RIPK1 INHIBITORS AND USE THEREOF GENZYME CORPORATION (US) 2026-03-18 EP claimed
WO-2025133915-A1 COMPOUNDS WHICH BIND TO PNPLA3I148M AND THEIR USE TO TREAT LIVER DISEASES NOVARTIS AG (CH) 2025-06-26 WO claimed
CN-119775930-A PMMA glue with high ionic conductivity and preparation method thereof 长园新能源材料研究院(广东)有限公司 2025-04-08 CN claimed
US-20250090501-A1 METHODS OF TREATING GUT MOTILITY DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-03-20 US claimed
WO-2024233544-A1 ISOXAZOLIDINES AS RIPK1 INHIBITORS AND USE THEREOF GENZYME CORPORATION (US) 2024-11-14 WO claimed
EP-4396630-A1 ELECTROACTIVE OPTICAL DEVICE PPG Industries Ohio Inc. (US) 2024-07-10 EP claimed
CN-114136941-B SARM1 enzyme inhibitor and screening method and application thereof 北京大学深圳研究生院 2024-04-16 CN claimed
CN-117695294-A Application of phenazopyridine hydrochloride in preparation of antibiotic reinforcing agent 中科帆凯(大连)新材料有限公司 2024-03-15 CN claimed
CN-116948220-A Preparation method of adjustable heterostructure low surface energy microsphere and preparation method of textile 浙江理工大学 2023-10-27 CN claimed
WO-2023130364-A1 METHOD FOR TESTING VIRUS CONTENT OF WATER ON THE BASIS OF ALUMINUM SALT COAGULATION PRETREATMENT 中国科学院生态环境研究中心 2023-07-13 WO claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
WO-2000021504-A1 ENCAPSULATION OF SENSITIVE LIQUID COMPONENTS INTO A MATRIX TO OBTAIN DISCRETE SHELF-STABLE PARTICLES GENERAL MILLS, INC. (US) 2000-04-20 WO claimed
EP-0935523-A4 EMBEDDING AND ENCAPSULATION OF CONTROLLED RELEASE PARTICLES GEN MILLS INC (US) 1999-12-29 EP claimed
EP-0935523-A1 EMBEDDING AND ENCAPSULATION OF CONTROLLED RELEASE PARTICLES GENERAL MILLS, INC. (US) 1999-08-18 EP claimed
WO-1998018610-A1 EMBEDDING AND ENCAPSULATION OF CONTROLLED RELEASE PARTICLES LENGERICH BERNHARD H VAN (US) 1998-05-07 WO claimed
EP-0741570-A1 METHOD FOR PREVENTING OR REDUCING PHOTOSENSITIVITY AND/OR PHOTOTOXICITY REACTIONS TO MEDICATIONS G.D. SEARLE & CO. (US) 1996-11-13 EP claimed
WO-1995020387-A1 METHOD FOR PREVENTING OR REDUCING PHOTOSENSITIVITY AND/OR PHOTOTOXICITY REACTIONS TO MEDICATIONS G.D. SEARLE & CO. (US) 1995-08-03 WO claimed
US-5357636-A Flexible protective medical gloves and methods for their use DRESDNER JR KARL P (US) 1994-10-25 US claimed
EP-0312132-B1 VETERINARY AND HUMAN MEDICAL REMEDY HAVING AN ANTIVIRAL AND ANTITUMOROUS ACTIVITY, CONTAINING 2,6-DIAMINO-3-PHENYL-AZO-PYRIDINE Hak, Barend Willem (NL) 1993-01-13 EP claimed
US-4056609-A Article for diagnosis of achlorhydria GUNN, KIRCHUBEL & MILLER (US) 1977-11-01 US claimed