SCHEMBL2649939

SCHEMBL2649939

NNC(=O)c1ccc(OS(=O)(=O)C(F)(F)F)c2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.43
CA2 P00918 2/20 0.40
CTSD P07339 2/20 0.40
CA1 P00915 1/20 0.40
CA9 Q16790 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGDS O60760 1/20 0.37
CDC25B P30305 1/20 0.36
NSD2 O96028 2/20 0.35
MITF O75030 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
NCOA1 Q15788 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
NCOA3 Q9Y6Q9 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4467822 0.82 PLK1 (0.44) PLK1CA2CA1CA9MEN1
SCHEMBL6851155 0.81 MEN1 (0.38) CA2CA1CA9MEN1KMT2A
SCHEMBL247360 0.77 CNR2 (0.55) MEN1KMT2ACDC25BGAAMAPT
SCHEMBL9470141 0.76 GPR3 (0.37) CA2CA1CA9MEN1KMT2A
SCHEMBL14400507 0.76 SLC2A1 (0.42) MEN1KMT2AGAACYP2C9SLC2A1
SCHEMBL466508 0.75 MAPT (0.52) PLK1CA2CTSDCA1CA9
SCHEMBL5891933 0.75 PLK1 (0.73) PLK1CTSDKMT2AALDH1A1KDM4E
SCHEMBL203899 0.74 MEN1 (0.42) MEN1KMT2AGAA
SCHEMBL29706003 0.74 MEN1 (0.42) MEN1KMT2AGAA
SCHEMBL8636736 0.73 IDO1 (0.46) PLK1ALDH1A1HPGDSCDC25BCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6613942-B1 Nonpeptide; 4-hydroxy benzoic acid hydrazides NOVO NORDISK A/S (DK) 2003-09-02 US disclosed
EP-0994848-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 2000-04-26 EP disclosed
WO-1999001423-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 1999-01-14 WO disclosed