SCHEMBL2650181

SCHEMBL2650181

N#Cc1cccnc1-n1ccccc1=O

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.46
RECQL P46063 1/20 0.46
DRD2 P14416 2/20 0.41
HTR2A P28223 1/20 0.41
ALDH1A1 P00352 2/20 0.40
MAPT P10636 1/20 0.40
HSD11B1 P28845 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
GRM1 Q13255 1/20 0.39
HDAC2 Q92769 1/20 0.38
KMT2A Q03164 1/20 0.38
PANK3 Q9H999 1/20 0.38
BCL6 P41182 1/20 0.38
ELANE P08246 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2658855 0.78 KDM4E (0.40) KDM4ERECQLDRD2HTR2AALDH1A1
SCHEMBL25427898 0.78 KDM4E (0.46) KDM4ERECQLDRD2HTR2AALDH1A1
SCHEMBL31247608 0.76 KDM4E (0.46) KDM4ERECQLDRD2HTR2AALDH1A1
SCHEMBL950862 0.76 ALDH1A1 (0.43) KDM4ERECQLDRD2HTR2AALDH1A1
SCHEMBL23754789 0.76 GRIN2D (0.42) KDM4EHSD11B1HDAC2CA12CA1
SCHEMBL27744470 0.75 KMT2A (0.49) KDM4EALDH1A1MAPTKMT2ACA12
SCHEMBL7130873 0.73 CYP2E1 (0.46) KDM4ERECQLDRD2HTR2AALDH1A1
SCHEMBL28417261 0.72 HSD11B1 (0.48) HSD11B1
SCHEMBL1882886 0.72 GRIA1 (0.45) KDM4EALDH1A1TDP1
SCHEMBL2918046 0.70 GRIA1 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003093273-A1 IMIDAZO-TRIAZINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 2003-11-13 WO disclosed