SCHEMBL7130873

SCHEMBL7130873

Cc1nccn1-c1ncccc1C#N

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2A6 P11509 1/20 0.46
ALDH1A1 P00352 3/20 0.44
MAPT P10636 1/20 0.44
HSD11B1 P28845 1/20 0.43
KDM4E B2RXH2 5/20 0.41
RECQL P46063 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
DRD2 P14416 5/20 0.39
HTR2A P28223 4/20 0.39
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ELANE P08246 2/20 0.38
HTR1A P08908 1/20 0.37
HTR7 P34969 1/20 0.37
GRM5 P41594 1/20 0.37
ICMT O60725 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26114212 0.79 KDM4E (0.46) CYP2E1CYP3A4CYP2A6ALDH1A1MAPT
SCHEMBL8501020 0.78 CYP3A4 (0.53) CYP2E1CYP3A4CYP2A6ALDH1A1MAPT
SCHEMBL8498623 0.75 CYP3A4 (0.50) CYP2E1CYP3A4CYP2A6ALDH1A1HSD11B1
SCHEMBL31247608 0.74 KDM4E (0.46) ALDH1A1MAPTHSD11B1KDM4ERECQL
SCHEMBL2650181 0.73 KDM4E (0.46) ALDH1A1MAPTHSD11B1KDM4ERECQL
SCHEMBL8502061 0.72 CYP3A4 (0.47) CYP2E1CYP3A4CYP2A6ALDH1A1RECQL
SCHEMBL8733365 0.72 CYP3A4 (0.47) CYP2E1CYP3A4CYP2A6ALDH1A1
SCHEMBL19080612 0.72 CYP3A4 (0.44) CYP2E1CYP3A4CYP2A6ALDH1A1
SCHEMBL3291168 0.71 KDM4E (0.50) ALDH1A1MAPTHSD11B1KDM4ERECQL
SCHEMBL950862 0.71 ALDH1A1 (0.43) ALDH1A1MAPTHSD11B1KDM4ERECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004043947-A1 NOVEL PYRIDINE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME LES LABORATOIRES SERVIER (FR) 2004-05-27 WO disclosed