SCHEMBL2650837

SCHEMBL2650837

[O]C(OCc1cccc(Cl)c1)c1cccc(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.51
CYP3A4 P08684 2/20 0.51
AGXT P21549 2/20 0.51
TACR1 P25103 2/20 0.48
MAOB P27338 4/20 0.44
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
RXRG P48443 1/20 0.43
HCAR2 Q8TDS4 1/20 0.43
PNMT P11086 2/20 0.43
FFAR1 O14842 1/20 0.42
MAOA P21397 2/20 0.42
TDO2 P48775 1/20 0.42
NR4A2 P43354 1/20 0.42
THRA P10827 1/20 0.42
THRB P10828 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6745046 0.89 CYP3A4 (0.50) IDO1CYP3A4AGXTTACR1MAOB
SCHEMBL6772852 0.76 MRGPRX4 (0.39)
SCHEMBL27606094 0.75 HDAC7 (0.42) IDO1
SCHEMBL10314841 0.75 CYP3A4 (0.58) IDO1CYP3A4AGXTTACR1MAOB
SCHEMBL2650976 0.74 FFAR1 (0.47) TACR1MAOBFFAR1MAOA
SCHEMBL2651208 0.74 IDO1 (0.54) IDO1AGXTMAOBFFAR1
SCHEMBL27625109 0.74 ACP3 (0.40) IDO1
SCHEMBL2651330 0.74 CYP3A4 (0.42) IDO1CYP3A4AGXTTACR1MAOB
SCHEMBL23164237 0.73 CYP3A4 (0.51) IDO1CYP3A4AGXTTACR1MAOB
SCHEMBL23163975 0.73 CYP3A4 (0.51) IDO1CYP3A4AGXTTACR1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1404335-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS Astrazeneca AB (SE) 2004-04-07 EP disclosed
WO-2003000267-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS ASTRAZENECA AB (SE) 2003-01-03 WO disclosed