SCHEMBL2651330

SCHEMBL2651330

N#Cc1ccccc1C([O])OCc1cccc(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.42
IDO1 P14902 2/20 0.42
AGXT P21549 2/20 0.42
GRM5 P41594 2/20 0.41
ALDH1A1 P00352 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CNR1 P21554 1/20 0.39
NR4A2 P43354 1/20 0.39
TACR1 P25103 2/20 0.38
MRGPRX4 Q96LA9 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2652312 0.85 GLA (0.45) GRM5TACR1MRGPRX4MAOAMAOB
SCHEMBL2650061 0.84 IDO1 (0.42) CYP3A4IDO1ALDH1A1KDM4EHSD17B10
SCHEMBL2651467 0.82 IDO1 (0.44) IDO1AGXTNPC1RAB9AMAOB
SCHEMBL2651154 0.81 MRGPRX4 (0.52) SMN1; SMN2MEN1KMT2ANPC1RAB9A
SCHEMBL2652010 0.77 IDO1 (0.40) IDO1KMT2ANPC1RAB9ANR4A2
SCHEMBL2652551 0.76 FFAR1 (0.41) ALDH1A1SMN1; SMN2KDM4EKMT2ATDP1
SCHEMBL2650837 0.74 IDO1 (0.51) CYP3A4IDO1AGXTNR4A2TACR1
SCHEMBL2650379 0.74 KAT6A (0.33) IDO1ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL6745046 0.73 CYP3A4 (0.50) CYP3A4IDO1AGXTNR4A2TACR1
SCHEMBL2650744 0.73 MAPK14 (0.37) ALDH1A1TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1404335-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS Astrazeneca AB (SE) 2004-04-07 EP disclosed
WO-2003000267-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS ASTRAZENECA AB (SE) 2003-01-03 WO disclosed