SCHEMBL2651

SCHEMBL2651

CCOC(=O)N(Cc1ccc(-c2ccccc2C#N)cc1)[C@H](C(=O)OCc1ccccc1)C(C)C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.52
LMNA P02545 1/20 0.52
POLB P06746 1/20 0.52
HSD17B10 Q99714 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
FFAR1 O14842 1/20 0.44
AKR1B1 P15121 1/20 0.44
OXTR P30559 1/20 0.41
AVPR1A P37288 1/20 0.41
AGTR1 P30556 4/20 0.41
PTPN1 P18031 1/20 0.40
LTB4R2 Q9NPC1 3/20 0.39
ABCB11 O95342 1/20 0.39
GP6 Q9HCN6 1/20 0.39
EGLN1 Q9GZT9 1/20 0.38
MME P08473 1/20 0.38
ESR2 Q92731 1/20 0.38
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
CTSS P25774 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1820 0.93 FFAR1 (0.43) ALDH1A1LMNAPOLBHSD17B10L3MBTL1
SCHEMBL3664 0.91 FFAR1 (0.45) ALDH1A1LMNAPOLBHSD17B10L3MBTL1
SCHEMBL2989 0.91 FFAR1 (0.43) ALDH1A1LMNAPOLBHSD17B10L3MBTL1
SCHEMBL6509546 0.89 ALDH1A1 (0.49) ALDH1A1LMNAPOLBHSD17B10L3MBTL1
SCHEMBL1809623 0.88 AGTR1 (0.54) FFAR1AKR1B1AGTR1LTB4R2ABCB11
SCHEMBL29378073 0.88 AGTR1 (0.54) FFAR1AKR1B1AGTR1LTB4R2ABCB11
SCHEMBL2140 0.88 AGTR1 (0.54) FFAR1AKR1B1AGTR1LTB4R2ABCB11
SCHEMBL3473572 0.88 FFAR1 (0.46) ALDH1A1LMNAPOLBHSD17B10L3MBTL1
SCHEMBL3473577 0.88 FFAR1 (0.46) ALDH1A1LMNAPOLBHSD17B10L3MBTL1
SCHEMBL2438545 0.86 FFAR1 (0.48) LMNAFFAR1AKR1B1OXTRAVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed