SCHEMBL2651293

SCHEMBL2651293

COc1cc(OCCBr)ccc1C=O

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.65
MAOB P27338 2/20 0.55
L3MBTL1 Q9Y468 1/20 0.48
CYP1A1 P04798 4/20 0.46
CYP1B1 Q16678 4/20 0.46
CYP1A2 P05177 3/20 0.46
TUBB1 Q9H4B7 1/20 0.46
ERN1 O75460 4/20 0.45
KDM4E B2RXH2 1/20 0.44
TSHR P16473 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
TRIM24 O15164 1/20 0.42
TYR P14679 1/20 0.42
TRIM33 Q9UPN9 1/20 0.42
MEN1 O00255 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
NFE2L2 Q16236 1/20 0.41
PRKDC P78527 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14397892 0.88 ALDH1A1 (0.65) ALDH1A1MAOBL3MBTL1CYP1A1CYP1B1
SCHEMBL31432675 0.88 ALDH1A1 (0.65) ALDH1A1MAOBL3MBTL1CYP1A1CYP1B1
SCHEMBL5143351 0.86 ALDH1A1 (0.67) ALDH1A1MAOBL3MBTL1CYP1A1CYP1B1
SCHEMBL20892596 0.86 ALDH1A1 (0.67) ALDH1A1MAOBL3MBTL1CYP1A1CYP1B1
SCHEMBL4059477 0.86 ALDH1A1 (0.67) ALDH1A1MAOBL3MBTL1CYP1A1CYP1B1
SCHEMBL18045690 0.86 ALDH1A1 (0.67) ALDH1A1MAOBL3MBTL1CYP1A1CYP1B1
SCHEMBL12344082 0.84 ALDH1A1 (0.65) ALDH1A1MAOBL3MBTL1CYP1A1CYP1B1
SCHEMBL2352641 0.84 ALDH1A1 (0.65) ALDH1A1MAOBL3MBTL1CYP1A1CYP1B1
SCHEMBL5654410 0.83 ALDH1A1 (0.63) ALDH1A1MAOBL3MBTL1CYP1A1CYP1B1
SCHEMBL5143349 0.83 ALDH1A1 (0.63) ALDH1A1MAOBL3MBTL1CYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6613942-B1 Nonpeptide; 4-hydroxy benzoic acid hydrazides NOVO NORDISK A/S (DK) 2003-09-02 US disclosed
EP-0994848-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 2000-04-26 EP disclosed
WO-1999001423-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 1999-01-14 WO disclosed
WO-1999001423-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 1999-01-14 WO disclosed