SCHEMBL2652010

SCHEMBL2652010

N#Cc1ccccc1C([O])OCc1ccccc1Cl

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.40
HSD11B1 P28845 2/20 0.39
FABP4 P15090 2/20 0.37
FABP5 Q01469 2/20 0.37
NR4A2 P43354 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
PGR P06401 1/20 0.35
CASP3 P42574 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
KMT2A Q03164 1/20 0.33
GAA P10253 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NPBWR1 P48145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2652551 0.88 FFAR1 (0.41) NPC1RAB9ACASP3SENP8SENP7
SCHEMBL2652111 0.84 IDO1 (0.41) IDO1NPC1RAB9AMAOB
SCHEMBL2650236 0.83 IDO1 (0.48) IDO1FABP4FABP5NR4A2NPC1
SCHEMBL2651003 0.83 IDO1 (0.40) IDO1NPC1RAB9AMAOBKMT2A
SCHEMBL2652007 0.83 TSHR (0.43) MAOBL3MBTL1
SCHEMBL2650110 0.80 TP53 (0.41) MAOBKMT2AGAA
SCHEMBL2651078 0.80 IDO1 (0.44) IDO1MAOAMAOBGAA
SCHEMBL2650879 0.79 ALDH1A1 (0.48) MAOBKMT2A
SCHEMBL2651330 0.77 CYP3A4 (0.42) IDO1NR4A2NPC1RAB9AMAOA
SCHEMBL2650744 0.76 MAPK14 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1404335-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS Astrazeneca AB (SE) 2004-04-07 EP disclosed
WO-2003000267-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS ASTRAZENECA AB (SE) 2003-01-03 WO disclosed