SCHEMBL2651467

SCHEMBL2651467

COc1cccc(COC([O])c2ccccc2C#N)c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.44
AGXT P21549 2/20 0.44
ABCB1 P08183 2/20 0.42
HTR1A P08908 2/20 0.42
DRD2 P14416 2/20 0.42
MAOB P27338 4/20 0.40
TAAR1 Q96RJ0 2/20 0.40
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
MMP13 P45452 1/20 0.39
CMA1 P23946 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2650061 0.85 IDO1 (0.42) IDO1MAOB
SCHEMBL2652312 0.83 GLA (0.45) MAOB
SCHEMBL2651330 0.82 CYP3A4 (0.42) IDO1AGXTMAOBRAB9ANPC1
SCHEMBL2651154 0.79 MRGPRX4 (0.52) RAB9ANPC1
SCHEMBL2651208 0.76 IDO1 (0.54) IDO1AGXTABCB1HTR1ADRD2
SCHEMBL2652551 0.74 FFAR1 (0.41) MAOBRAB9ANPC1
SCHEMBL11118935 0.73 ABCB1 (0.58) ABCB1HTR1ADRD2TAAR1
SCHEMBL2652007 0.72 TSHR (0.43) MAOB
SCHEMBL2650379 0.72 KAT6A (0.33) IDO1
SCHEMBL17217219 0.72 IDO1 (0.47) IDO1AGXTABCB1HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1404335-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS Astrazeneca AB (SE) 2004-04-07 EP disclosed
WO-2003000267-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS ASTRAZENECA AB (SE) 2003-01-03 WO disclosed