SCHEMBL26523562

SCHEMBL26523562

NC(=O)C12CC1N(c1cccc(Cl)n1)C2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 3/20 0.40
HTR3B O95264 3/20 0.40
HTR3A P46098 3/20 0.40
HTR3D Q70Z44 3/20 0.40
HTR3C Q8WXA8 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
NFKB1 P19838 1/20 0.40
ALDH1A1 P00352 4/20 0.36
ALOX5 P09917 2/20 0.35
GAA P10253 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
GPX4 P36969 1/20 0.33
MGLL Q99685 1/20 0.33
CHRM4 P08173 2/20 0.32
GRM4 Q14833 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4234258 0.68 HTR3E (0.42) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL31141160 0.64 HTR3E (0.40) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL21723552 0.64 KMT2A (0.46) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL21723551 0.64 KMT2A (0.46) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL28552581 0.63 ADORA2A (0.45) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL20202159 0.62 HTR3E (0.43) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL9005356 0.62 KMT2A (0.50) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL2828415 0.62 ALDH1A1 (0.50) ALOX15TSHRALDH1A1GAAKDM4E
SCHEMBL25384299 0.61 GAA (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL28934391 0.61 GAA (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023187677-A1 N-(PYRROLIDIN-3-YL OR PIPERIDIN-4-YL)ACETAMIDE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-10-05 WO disclosed