SCHEMBL2652485

SCHEMBL2652485

N#Cc1c(F)cc(N)cc1-c1ccccc1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
KDM4E B2RXH2 2/20 0.49
GLA P06280 1/20 0.49
GAA P10253 1/20 0.49
HPGD P15428 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
ADORA1 P30542 8/20 0.47
ADORA2A P29274 7/20 0.47
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
ADORA2B P29275 3/20 0.38
TRPV4 Q9HBA0 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
CUL4A Q13619 1/20 0.36
CHUK O15111 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2648001 0.78 ADORA1 (0.42) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL2569036 0.77 ADORA1 (0.46) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL1947934 0.77 TRPV4 (0.58) KDM4EGAAADORA1ADORA2AADORA2B
SCHEMBL2650355 0.76 CYP11B1 (0.46) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL30415829 0.74 CYP11B1 (0.50) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL13614777 0.74 CYP11B1 (0.50) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL2650101 0.72 ADORA1 (0.47) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL6251132 0.72 KDM4E (0.77) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL25260661 0.71 BRD4 (0.51) ALDH1A1KDM4EHPGDSMN1; SMN2ADORA2A
SCHEMBL27091735 0.71 ALDH1A1 (0.48) ALDH1A1KDM4EGLAGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1381606-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 2004-01-21 EP disclosed
WO-2002074773-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 2002-09-26 WO disclosed