SCHEMBL2650101

SCHEMBL2650101

N#Cc1c(-c2ccccc2F)ccc(N)c1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.47
ADORA2A P29274 4/20 0.47
ALDH1A1 P00352 5/20 0.43
KDM4E B2RXH2 3/20 0.43
GAA P10253 2/20 0.43
HPGD P15428 2/20 0.43
GLA P06280 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 2/20 0.39
MAPK1 P28482 1/20 0.39
DYRK1A Q13627 2/20 0.39
ADORA2B P29275 2/20 0.38
CUL4A Q13619 1/20 0.36
CHUK O15111 1/20 0.36
LRRK2 Q5S007 1/20 0.36
EEF2K O00418 1/20 0.35
GRIA2 P42262 1/20 0.34
GRIA4 P48058 1/20 0.34
MPL P40238 1/20 0.34
GABRG2 P18507 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6695094 0.79 ADORA1 (0.40) ADORA1ADORA2AALDH1A1KDM4EGAA
SCHEMBL21199975 0.77 MPL (0.44) ADORA1ADORA2AALDH1A1KDM4EDYRK1A
SCHEMBL2569036 0.77 ADORA1 (0.46) ADORA1ADORA2AALDH1A1KDM4EGAA
SCHEMBL29906554 0.75 TRPV4 (0.37) ADORA1ADORA2AALDH1A1KDM4EGAA
SCHEMBL2597730 0.75 TRPV4 (0.37) ADORA1ADORA2AALDH1A1KDM4EGAA
SCHEMBL2651221 0.75 CYP11B1 (0.41) ADORA1ADORA2AALDH1A1KDM4EGAA
SCHEMBL2651898 0.74 ADORA1 (0.41) ADORA1ADORA2AALDH1A1KDM4EGAA
SCHEMBL27886232 0.73 ALDH1A1 (0.53) ADORA1ADORA2AALDH1A1KDM4EGAA
SCHEMBL2652485 0.72 ALDH1A1 (0.49) ADORA1ADORA2AALDH1A1KDM4EGAA
SCHEMBL28456456 0.72 MPL (0.43) ADORA1ADORA2AALDH1A1KDM4EDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002074772-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 2002-09-26 WO disclosed