SCHEMBL2652913

SCHEMBL2652913

N#Cc1c(-c2ccccc2)ccc(Br)c1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.46
L3MBTL1 Q9Y468 3/20 0.46
KDM4E B2RXH2 5/20 0.43
HPGD P15428 5/20 0.43
NPSR1 Q6W5P4 2/20 0.43
RXFP1 Q9HBX9 1/20 0.43
ALDH1A1 P00352 6/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
ADORA2A P29274 6/20 0.40
ADORA1 P30542 6/20 0.40
PPARG P37231 1/20 0.40
NCOA2 Q15596 1/20 0.40
NCOA1 Q15788 1/20 0.40
NCOA3 Q9Y6Q9 1/20 0.40
SQOR Q9Y6N5 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29967703 1.00 MAPK1 (0.46) MAPK1L3MBTL1KDM4EHPGDNPSR1
SCHEMBL2569037 0.81 ALDH1A1 (0.44) MAPK1L3MBTL1KDM4EHPGDNPSR1
SCHEMBL6695094 0.81 ADORA1 (0.40) MAPK1KDM4EHPGDNPSR1RXFP1
SCHEMBL16122421 0.80 ALDH1A1 (0.42) MAPK1L3MBTL1KDM4EHPGDNPSR1
SCHEMBL28871241 0.79 ALDH1A1 (0.43) MAPK1L3MBTL1KDM4EHPGDALDH1A1
SCHEMBL421377 0.79 ALDH1A1 (0.41) MAPK1L3MBTL1KDM4EHPGDNPSR1
SCHEMBL9854261 0.78 SQOR (0.40) MAPK1L3MBTL1KDM4EHPGDNPSR1
SCHEMBL4958212 0.78 ALDH1A1 (0.53) MAPK1L3MBTL1KDM4EHPGDNPSR1
SCHEMBL16122425 0.77 ADORA1 (0.51) MAPK1L3MBTL1KDM4EHPGDNPSR1
SCHEMBL29052685 0.77 ADORA1 (0.49) MAPK1L3MBTL1KDM4EHPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed
EP-1381606-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 2004-01-21 EP disclosed
WO-2002074773-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 2002-09-26 WO disclosed