SCHEMBL2654541

SCHEMBL2654541

CCOC(=O)Cc1csc(N)n1.CCOC(=O)Cc1csc(NC(=O)C(CC2CCCC2)c2ccc(-c3cccc4ccccc34)cc2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTC4S Q16873 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.46
ALDH1A1 P00352 4/20 0.45
TDP1 Q9NUW8 1/20 0.45
GCK P35557 2/20 0.43
LMNA P02545 3/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
GALR3 O60755 1/20 0.42
POLB P06746 2/20 0.42
GAA P10253 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2648137 0.96 LTC4S (0.52) LTC4SSMN1; SMN2ALDH1A1TDP1GCK
SCHEMBL2647572 0.89 GCK (0.46) LTC4SSMN1; SMN2GCKTP53NPC1
SCHEMBL6596927 0.88 ALDH1A1 (0.49) SMN1; SMN2ALDH1A1TDP1GCKLMNA
SCHEMBL2648107 0.86 ALDH1A1 (0.56) SMN1; SMN2ALDH1A1TDP1GCKLMNA
SCHEMBL2647650 0.84 GCK (0.48) GCK
SCHEMBL2647253 0.83 ALDH1A1 (0.54) SMN1; SMN2ALDH1A1TDP1GCKLMNA
SCHEMBL2648600 0.83 GCK (0.47) GCK
SCHEMBL2647614 0.82 GCK (0.49) GCK
SCHEMBL2646210 0.81 MAPT (0.59) SMN1; SMN2ALDH1A1TDP1GCKLMNA
SCHEMBL2656498 0.80 ALDH1A1 (0.49) SMN1; SMN2ALDH1A1TDP1GCKLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1282611-A1 SUBSTITUTED PHENYLACETAMIDES AND THEIR USE AS GLUCOKINASE ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2003-02-12 EP disclosed
WO-2001085706-A1 SUBSTITUTED PHENYLACETAMIDES AND THEIR USE AS GLUCOKINASE ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2001-11-15 WO disclosed