SCHEMBL2654639

SCHEMBL2654639

CCOC(=O)c1ccc(CCc2cc(Br)ccc2O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
CYP1A2 P05177 2/20 0.56
CYP3A4 P08684 2/20 0.56
HPGD P15428 2/20 0.56
TP53 P04637 1/20 0.56
CYP2C9 P11712 1/20 0.56
ALOX15 P16050 1/20 0.56
ALOX12 P18054 1/20 0.56
CYP2C19 P33261 1/20 0.56
CKS1B P61024 1/20 0.56
SKP2 Q13309 1/20 0.56
HIF1A Q16665 1/20 0.56
HSD17B10 Q99714 1/20 0.56
CCR6 P51684 1/20 0.54
HKDC1 Q2TB90 1/20 0.54
CA12 O43570 2/20 0.52
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
CA7 P43166 2/20 0.52
CA9 Q16790 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14130672 0.88 CA12 (0.54) ALDH1A1CYP1A2CYP3A4HPGDCA12
SCHEMBL6274539 0.84 HPGD (0.56) ALDH1A1CYP1A2CYP3A4HPGDTP53
SCHEMBL16687963 0.81 CA12 (0.58) ALDH1A1CYP1A2CYP3A4HPGDTP53
SCHEMBL8409449 0.81 CA12 (0.59) ALDH1A1CYP1A2CYP3A4HPGDTP53
SCHEMBL11252769 0.80 HKDC1 (0.60) ALDH1A1ALOX15CKS1BSKP2HSD17B10
SCHEMBL12199135 0.80 CA1 (0.68) ALDH1A1CYP1A2CYP3A4HPGDCA12
SCHEMBL8326087 0.79 ALDH1A1 (0.64) ALDH1A1CYP1A2CYP3A4HPGDTP53
SCHEMBL274513 0.76 CA1 (0.68) ALDH1A1CYP1A2CYP3A4HPGDCA12
SCHEMBL6274720 0.76 CCR6 (0.48) ALDH1A1CYP1A2CYP3A4HPGDTP53
SCHEMBL1515780 0.76 CA12 (0.68) ALDH1A1CYP1A2CYP3A4HPGDTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863755-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES Merck & Co., Inc. (US) 2007-12-12 EP disclosed
WO-2006102067-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES MERCK & CO., INC. (US) 2006-09-28 WO disclosed