SCHEMBL2655552

SCHEMBL2655552

CCCCOc1cc(C(=O)Nc2ncc(C(=O)O)s2)c2ccccc2n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
KDM4E B2RXH2 2/20 0.57
HPGD P15428 2/20 0.57
ABCB11 O95342 1/20 0.57
LMNA P02545 1/20 0.57
CYP1A2 P05177 1/20 0.57
GAA P10253 1/20 0.57
CYP2D6 P10635 1/20 0.57
SCN1A P35498 1/20 0.57
OPRK1 P41145 1/20 0.57
KCNH2 Q12809 1/20 0.57
CACNA1C Q13936 1/20 0.57
SCN5A Q14524 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
GHSR Q92847 1/20 0.57
SCN2A Q99250 1/20 0.57
SCN3A Q9NY46 1/20 0.57
ALOX15 P16050 1/20 0.56
HTT P42858 1/20 0.56
NR2E1 Q9Y466 4/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2655547 0.85 ALDH1A1 (0.52) ALDH1A1KDM4EHPGDLMNAGAA
SCHEMBL2654506 0.82 ALDH1A1 (0.48) ALDH1A1KDM4EHPGDLMNAHTT
SCHEMBL6250517 0.79 KDM4E (0.65) ALDH1A1KDM4EHPGDABCB11LMNA
SCHEMBL31673005 0.79 KDM4E (0.65) ALDH1A1KDM4EHPGDABCB11LMNA
SCHEMBL4678263 0.79 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDLMNAGAA
SCHEMBL31729873 0.76 NR2E1 (0.67) ALDH1A1KDM4EHPGDABCB11LMNA
SCHEMBL9198147 0.76 HTR3E (0.61) ALDH1A1KDM4EHPGDABCB11LMNA
SCHEMBL4677599 0.76 ALDH1A1 (0.48) ALDH1A1KDM4EHPGDLMNASMN1; SMN2
SCHEMBL9198080 0.75 HTR3E (0.61) ALDH1A1KDM4EHPGDABCB11LMNA
SCHEMBL28378761 0.75 KDM4E (0.62) ALDH1A1KDM4EHPGDABCB11LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583532-A1 QUINOLINE DERIVATIVES AS GLUCOKINASE LIGANDS Astrazeneca AB (SE) 2005-10-12 EP claimed
WO-2004045614-A1 QUINOLINE DERIVATIVES AS GLUCOKINASE LIGANDS ASTRAZENECA AB (SE) 2004-06-03 WO claimed
EP-1583532-A1 QUINOLINE DERIVATIVES AS GLUCOKINASE LIGANDS Astrazeneca AB (SE) 2005-10-12 EP disclosed
WO-2004045614-A1 QUINOLINE DERIVATIVES AS GLUCOKINASE LIGANDS ASTRAZENECA AB (SE) 2004-06-03 WO disclosed