SCHEMBL2657525

SCHEMBL2657525

C[C@@H](N)c1ccc2c(c1)ncn2-c1cccc(-c2cc(C#N)ccc2Cl)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36
GABRA4 P48169 1/20 0.36
GABRE P78334 1/20 0.36
GABRA6 Q16445 1/20 0.36
GABRG1 Q8N1C3 1/20 0.36
GABRG3 Q99928 1/20 0.36
GABRQ Q9UN88 1/20 0.36
LCK P06239 5/20 0.35
IRAK4 Q9NWZ3 3/20 0.35
JAK2 O60674 4/20 0.35
JAK3 P52333 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2658638 0.86 LCK (0.35) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL2655702 0.85 LCK (0.40) LCKIRAK4FGFR1ROCK1CDK2
SCHEMBL2657774 0.85 JAK2 (0.43) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL2656663 0.83 GABRA1 (0.43) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1615749 0.82 GABRA1 (0.46) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL1617069 0.82 GABRA1 (0.46) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL2657634 0.81 GABRA1 (0.49) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL2669851 0.73 LCK (0.43) LCKIRAK4FGFR1ROCK1
SCHEMBL1762063 0.73 GABRA1 (0.48) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL1762117 0.73 GABRA1 (0.48) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010055126-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE FOR MODULATING THE GABAA RECEPTOR COMPLEX NEUROSEARCH A/S (DK) 2010-05-20 WO claimed
WO-2010055126-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE FOR MODULATING THE GABAA RECEPTOR COMPLEX NEUROSEARCH A/S (DK) 2010-05-20 WO disclosed