SCHEMBL2657774

SCHEMBL2657774

C[C@@H](N)c1ccc2c(c1)ncn2-c1cccc(-c2cccc(C#N)c2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.43
JAK3 P52333 3/20 0.43
LCK P06239 4/20 0.41
GRM5 P41594 4/20 0.39
GRM2 Q14416 1/20 0.39
MET P08581 1/20 0.38
PDE1A P54750 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE1C Q14123 1/20 0.38
PDE3A Q14432 1/20 0.38
PDE11A Q9HCR9 1/20 0.38
PDE10A Q9Y233 1/20 0.38
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRB1 P18505 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2657525 0.85 GABRP (0.36) JAK2JAK3LCKMETGABRP
SCHEMBL2656663 0.82 GABRA1 (0.43) LCKGRM2METGABRA1GABRG2
SCHEMBL2659136 0.80 GABRA1 (0.55) JAK2JAK3GRM5GRM2GABRP
SCHEMBL2658638 0.80 LCK (0.35) LCKGABRA1GABRG2GABRB3GABRA5
SCHEMBL2655702 0.76 LCK (0.40) LCKCDK2IRAK4
SCHEMBL2669851 0.76 LCK (0.43) LCKIRAK4
SCHEMBL1615749 0.74 GABRA1 (0.46) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL1617069 0.74 GABRA1 (0.46) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL1616646 0.71 GABRA1 (0.66) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1616062 0.71 GABRA1 (0.66) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010055126-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE FOR MODULATING THE GABAA RECEPTOR COMPLEX NEUROSEARCH A/S (DK) 2010-05-20 WO claimed
WO-2010055126-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE FOR MODULATING THE GABAA RECEPTOR COMPLEX NEUROSEARCH A/S (DK) 2010-05-20 WO disclosed