SCHEMBL2659102

SCHEMBL2659102

CCOC(=O)c1cc2ccc(Cl)c(NS(=O)(=O)c3sccc3C)c2[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.48
CCNB1 P14635 1/20 0.48
ALOX15 P16050 1/20 0.45
MMP13 P45452 4/20 0.43
MMP2 P08253 3/20 0.43
ALDH1A1 P00352 6/20 0.39
KDM4E B2RXH2 5/20 0.39
HPGD P15428 4/20 0.39
RAB9A P51151 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
HSD17B10 Q99714 1/20 0.39
MAPT P10636 5/20 0.38
LMNA P02545 4/20 0.38
NPC1 O15118 3/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
GAA P10253 2/20 0.38
GLA P06280 1/20 0.38
ATM Q13315 1/20 0.38
LGALS8 O00214 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2659861 0.88 DAO (0.39) CDK1CCNB1ALDH1A1HPGDHSD17B10
SCHEMBL2660574 0.87 CDK1 (0.33) CDK1CCNB1KDM4EMAPTLMNA
SCHEMBL1653270 0.85 CDK1 (0.50) CDK1CCNB1ALOX15MMP13MMP2
SCHEMBL2660262 0.84 PPIA (0.32) CDK1CCNB1LGALS8LGALS3
SCHEMBL2659960 0.81 KDM4E (0.45) CDK1CCNB1ALOX15MMP13MMP2
SCHEMBL1653957 0.77 MEN1 (0.48) CDK1CCNB1ALOX15MMP13MMP2
SCHEMBL2660539 0.76 MMP13 (0.40) CDK1CCNB1ALOX15MMP13MMP2
SCHEMBL2660569 0.75 ALDH1A1 (0.39) CDK1CCNB1ALOX15MMP13MMP2
SCHEMBL30525398 0.74 CDK1 (0.64) CDK1CCNB1ALOX15MMP13MMP2
SCHEMBL4048527 0.74 CDK1 (0.64) CDK1CCNB1ALOX15MMP13MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074119-A1 INDOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008050821-A1 INDOLE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-02 WO disclosed