SCHEMBL2659423

SCHEMBL2659423

Cc1ccsc1S(=O)(=O)Nc1cccc2cc(C(=O)NCC(C)(CN3CCN(C(=O)O)CC3)SCc3ccccc3)[nH]c12

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 3/20 0.32
PKM P14618 1/20 0.32
NSD2 O96028 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
PLCG2 P16885 1/20 0.31
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30
THRB P10828 1/20 0.30
MAPT P10636 1/20 0.30
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2660564 0.92 KDM4E (0.37) LMNAMAPT
SCHEMBL2661515 0.89 MAPK8 (0.33) LMNATP53MAPT
SCHEMBL2659227 0.86 NSD2 (0.35) NSD2HDAC3HDAC1PLCG2MAPT
SCHEMBL2659015 0.85 HDAC3 (0.32) HRH4PKMNSD2HDAC3HDAC1
SCHEMBL2659696 0.84 NSD2 (0.37) NSD2HDAC3HDAC1PLCG2MAPT
SCHEMBL2659433 0.83 NSD2 (0.33) HRH4NSD2HDAC3HDAC1PLCG2
SCHEMBL2659093 0.82 NSD2 (0.36) NSD2HDAC3HDAC1PLCG2MAPT
SCHEMBL2659972 0.81 MCL1 (0.33) NSD2HDAC3HDAC1PLCG2LMNA
SCHEMBL2659077 0.81 NSD2 (0.33) NSD2HDAC3HDAC1PLCG2LMNA
SCHEMBL2659425 0.80 SMN1; SMN2 (0.35) PKMPLCG2LMNATP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074119-A1 INDOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008050821-A1 INDOLE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-02 WO disclosed