SCHEMBL2659639

SCHEMBL2659639

CCOC(=O)c1cc2cccc(NS(=O)(=O)c3nc(C)cn3C)c2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.45
CCNB1 P14635 1/20 0.45
KMT2A Q03164 4/20 0.42
MEN1 O00255 2/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
LMNA P02545 2/20 0.42
NPC1 O15118 1/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
ATM Q13315 1/20 0.42
MMP2 P08253 4/20 0.42
MMP13 P45452 4/20 0.42
POLB P06746 2/20 0.42
MMP14 P50281 2/20 0.40
BRD4 O60885 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2659829 0.88 ALDH1A1 (0.39) KMT2AMEN1ALDH1A1HPGDMMP2
SCHEMBL1653148 0.81 MMP2 (0.59) CDK1CCNB1KMT2AMEN1KDM4E
SCHEMBL2661679 0.81 KMT2A (0.38) CDK1CCNB1KMT2AMEN1KDM4E
SCHEMBL1653146 0.81 LMNA (0.60) CDK1CCNB1KMT2AMEN1KDM4E
SCHEMBL1653519 0.80 TSHR (0.48) CDK1CCNB1KMT2AMEN1KDM4E
SCHEMBL12783421 0.79 CDK1 (0.46) CDK1CCNB1KMT2AMEN1KDM4E
SCHEMBL2659240 0.78 POLB (0.50) CDK1CCNB1KMT2AMEN1KDM4E
SCHEMBL1653127 0.78 MAPT (0.51) CDK1CCNB1KMT2AMEN1KDM4E
SCHEMBL1653948 0.78 ALDH1A1 (0.52) CDK1CCNB1KMT2AMEN1KDM4E
SCHEMBL14601687 0.78 LMNA (0.48) CDK1CCNB1KMT2AMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074119-A1 INDOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008050821-A1 INDOLE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-02 WO disclosed