SCHEMBL2660481

SCHEMBL2660481

C=[C]C(=O)NCC1CCN(C)CC1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
MAPT P10636 1/20 0.40
NAMPT P43490 4/20 0.40
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC4 P56524 1/20 0.37
GSK3B P49841 1/20 0.37
HDAC3 O15379 3/20 0.37
HDAC8 Q9BY41 3/20 0.37
EPHX1 P07099 2/20 0.36
EPHX2 P34913 2/20 0.36
PARP1 P09874 1/20 0.35
MAP4K4 O95819 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13621194 0.80 TDP1 (0.67) NCF1TDP1MAPTNAMPTHDAC1
SCHEMBL8136269 0.78 MTNR1A (0.45) NCF1TDP1MAPTNAMPTHDAC4
SCHEMBL16494745 0.78 CYP2D6 (0.50) NCF1TDP1MAPTNAMPTHDAC1
SCHEMBL21730499 0.78 MAPT (0.38) NCF1TDP1MAPTNAMPTHDAC1
SCHEMBL23173065 0.77 MAPT (0.43) NCF1TDP1MAPTNAMPTHDAC1
SCHEMBL20711077 0.76 TGM2 (0.41) NCF1TDP1MAPTNAMPTHDAC4
SCHEMBL24239177 0.76 TDP1 (0.50) NCF1TDP1MAPTNAMPTHDAC1
SCHEMBL13853539 0.75 MAPT (0.48) NCF1TDP1MAPTNAMPTHDAC1
SCHEMBL12935918 0.75 CKS1B (0.45) NCF1TDP1MAPTNAMPTHDAC1
SCHEMBL12964152 0.75 CKS1B (0.46) NCF1TDP1MAPTNAMPTHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678144-A1 1,5,7-TRISUBSTITUTED BENZIMIDAZOLE DERIVATIVES AND THEIR USE FOR MODULATING THE GABA-a RECEPTOR COMPLEX Akzo Nobel N.V. (NL) 2006-07-12 EP disclosed
WO-2005040131-A1 1,5,7-TRISUBSTITUTED BENZIMIDAZOLE DERIVATIVES AND THEIR USE FOR MODULATING THE GABAA RECEPTOR COMPLEX AKZO NOBEL N.V. (NL) 2005-05-06 WO disclosed