SCHEMBL2661069

SCHEMBL2661069

COCCOc1cc(NS(=O)(=O)c2sccc2C)c2[nH]c(C(N)=O)cc2c1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.32
CHEK1 O14757 3/20 0.32
CHEK2 O96017 2/20 0.32
USP2 O75604 1/20 0.32
USP8 P40818 1/20 0.32
ITGB3 P05106 1/20 0.32
ITGAV P06756 1/20 0.32
MCL1 Q07820 1/20 0.31
MEN1 O00255 3/20 0.31
KMT2A Q03164 3/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31
CNKSR1 Q969H4 1/20 0.31
LGALS8 O00214 1/20 0.30
LGALS3 P17931 1/20 0.30
HPGD P15428 1/20 0.30
MAPT P10636 1/20 0.30
SYK P43405 1/20 0.30
BRAF P15056 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2661084 0.92 MCL1 (0.33) PIK3CAUSP2USP8ITGB3ITGAV
SCHEMBL2660569 0.90 ALDH1A1 (0.39) MEN1KMT2AALDH1A1POLBGAA
SCHEMBL2660500 0.84 KDM4E (0.36) MCL1MEN1KMT2AGAALGALS8
SCHEMBL2660266 0.83 MEN1 (0.39) MEN1KMT2AALDH1A1POLBMAPT
SCHEMBL2659586 0.81 MAPT (0.36) CHEK1CHEK2MCL1MEN1KMT2A
SCHEMBL2660294 0.79 NSD2 (0.37) MEN1KMT2A
SCHEMBL2660059 0.78 ALDH1A1 (0.46) USP2USP8MEN1KMT2AALDH1A1
SCHEMBL2660342 0.77
SCHEMBL2660539 0.76 MMP13 (0.40) MEN1KMT2AALDH1A1GAALGALS8
SCHEMBL2659681 0.75 SLC40A1 (0.37) MCL1KMT2AGAALGALS8LGALS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074119-A1 INDOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008050821-A1 INDOLE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-02 WO disclosed