SCHEMBL2661997

SCHEMBL2661997

Cc1ccc(NC(=O)Nc2ncc(CC(=O)OC(C(N)=O)c3cnc(NC(=O)Nc4ccc(C)cc4OCC(C)C)s3)s2)c(OCC(C)C)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
TSHR P16473 1/20 0.36
CCNE1 P24864 3/20 0.35
CDK2 P24941 3/20 0.35
CDK5 Q00535 3/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
LPAR1 Q92633 2/20 0.34
SMN1; SMN2 Q16637 3/20 0.33
POLB P06746 1/20 0.33
CCNT1 O60563 1/20 0.32
CDK1 P06493 1/20 0.32
CDK4 P11802 1/20 0.32
CCNB1 P14635 1/20 0.32
CCNA2 P20248 1/20 0.32
CCND1 P24385 1/20 0.32
CDK7 P50613 1/20 0.32
CDK9 P50750 1/20 0.32
CCNH P51946 1/20 0.32
MNAT1 P51948 1/20 0.32
CDK5R1 Q15078 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1343187 0.86 LPAR1 (0.39) ALDH1A1TSHRL3MBTL1LPAR1SMN1; SMN2
SCHEMBL1342497 0.83 ITGB1 (0.42) ALDH1A1TSHRCCNE1CDK2CDK5
SCHEMBL2661995 0.83 ITGB1 (0.39) ALDH1A1TSHRCCNE1CDK2CDK5
SCHEMBL1342668 0.82 LPAR1 (0.39) ALDH1A1TSHRL3MBTL1LPAR1SMN1; SMN2
SCHEMBL2649815 0.82 POLB (0.40) ALDH1A1TSHRL3MBTL1SMN1; SMN2POLB
SCHEMBL1343714 0.81 LPAR1 (0.38) L3MBTL1LPAR1SMN1; SMN2MAPK14MAPK13
SCHEMBL1340994 0.80 LPAR1 (0.36) ALDH1A1TSHRLPAR1SMN1; SMN2MYC
SCHEMBL6695210 0.80 CCNE1 (0.39) ALDH1A1CCNE1CDK2CDK5LPAR1
SCHEMBL1343242 0.79 LPAR1 (0.37) L3MBTL1LPAR1SMN1; SMN2POLBMAPK14
SCHEMBL6695295 0.79 AURKA (0.40) CDK2LPAR1MAPK14AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1531815-A1 GLUCOKINASE ACTIVATORS NOVO NORDISK A/S (DK) 2005-05-25 EP disclosed
WO-2004002481-A1 ARYL CARBONYL DERIVATIVES AS THERAPEUTIC AGENTS NOVO NORDISK A/S (DK) 2004-01-08 WO disclosed