SCHEMBL266416

SCHEMBL266416

CC(N)Cc1ccccc1O

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.50
TAAR1 Q96RJ0 3/20 0.50
SLC6A4 P31645 2/20 0.50
SLC6A3 Q01959 2/20 0.50
ADRB1 P08588 1/20 0.50
HTR1A P08908 1/20 0.50
ADRA2A P08913 1/20 0.50
HTR1D P28221 1/20 0.50
HTR1B P28222 1/20 0.50
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
HTR1E P28566 1/20 0.50
HTR7 P34969 1/20 0.50
HTR2B P41595 1/20 0.50
HTR6 P50406 1/20 0.50
MAOA P21397 1/20 0.50
HSPA5 P11021 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
CYP2A6 P11509 1/20 0.50
ADORA2A P29274 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4742791 1.00 SLC6A2 (0.50) SLC6A2TAAR1SLC6A4SLC6A3ADRB1
SCHEMBL5914402 1.00 SLC6A2 (0.50) SLC6A2TAAR1SLC6A4SLC6A3ADRB1
Hydrochloric Acid SCHEMBL724080 0.98 SLC6A2 (0.49) SLC6A2TAAR1SLC6A4SLC6A3ADRB1
Bromide SCHEMBL6052803 0.98 SLC6A2 (0.49) SLC6A2TAAR1SLC6A4SLC6A3ADRB1
Iodide SCHEMBL6052802 0.98 SLC6A2 (0.49) SLC6A2TAAR1SLC6A4SLC6A3ADRB1
SCHEMBL2857779 0.84 SLC6A2 (0.61) SLC6A2TAAR1SLC6A4SLC6A3ADRB1
SCHEMBL19971988 0.83 CYP2D6 (0.47) SLC6A2TAAR1SLC6A4SLC6A3HSPA5
SCHEMBL632694 0.83 GABRA1 (0.55) SLC6A2TAAR1SLC6A4SLC6A3MAOA
SCHEMBL108067 0.82 GABRA1 (0.64) TAAR1HSPA5
SCHEMBL3071437 0.82 HSPA5 (0.54) SLC6A2TAAR1SLC6A4SLC6A3HSPA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 139 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3870170-B1 TREATMENT OF PRESBYOPIA AND MYDRIASIS WITH PHENTOLAMINE OPUS GENETICS INC (US) 2026-02-25 EP claimed
EP-3413872-B1 NON-INVASIVE OCULAR DRUG DELIVERY INSERT TECHNOLOGY UNIV DE COIMBRA (PT) 2024-10-02 EP claimed
EP-2991621-B1 TWO-LAYER OCULAR IMPLANT RETINA FOUND OF THE SOUTHWEST (US) 2020-12-09 EP claimed
EP-2884962-B1 PREPARATION OF DESICCATED LIPOSOMES FOR USE IN COMPRESSIBLE DELIVERY SYSTEMS SMARTEK INT LLC (US) 2019-05-01 EP claimed
US-9757376-B2 Pharmaceutical compositions GM PHARMACEUTICALS, INC. (US) 2017-09-12 US claimed
CN-104277043-B One-dimensional organic semiconductor nanotube and its preparation method and application INSTITUTE OF CHEMISTRY, CHINESE ACADEMY OF SCIENCES (CN) 2017-01-04 CN claimed
EP-2493459-B1 OCULAR DRUG DELIVERY DEVICES ATON PHARMA INC (US) 2016-08-24 EP claimed
EP-2991621-A2 TWO-LAYER OCULAR IMPLANT Odin Biotech (US) 2016-03-09 EP claimed
EP-1825851-B1 Combination therapy for effecting weight loss and treating obesity VIVUS INC (US) 2015-07-22 EP claimed
EP-2305227-B1 Combination therapy for the treatment of diabetes associated with obesity VIVUS INC (US) 2015-05-06 EP claimed
EP-2352459-A1 MACROCYCLIC LACTONE COMPOUNDS AND METHODS FOR THEIR USE Elixir Medical Corporation (US) 2011-08-10 EP claimed
EP-1671624-B1 Delivery device for a controlled drug release of an active agent into the posterior section of the eye SURMODICS INC (US) 2010-08-11 EP claimed
WO-2010040064-A1 MACROCYCLIC LACTONE COMPOUNDS AND METHODS FOR THEIR USE ELIXIR MEDICAL CORPORATION (US) 2010-04-08 WO claimed
EP-1276462-B1 SUSTAINED RELEASE DRUG DELIVERY DEVICES, METHODS OF USE, AND METHODS OF MANUFACTURING THEREOF PSIVIDA INC (US) 2008-09-24 EP claimed
EP-1187603-B1 COMBINATION THERAPY FOR EFFECTING WEIGHT LOSS AND TREATING OBESITY VIVUS INC (US) 2007-08-08 EP claimed
CN-1703199-A Aggregate with enhanced deformability comprising at least three amphiphiles for improved transport through a semi-permeable barrier and use of non-invasive drugs in vivo, in particular through the skin IDEA AG (DE) 2005-11-30 CN claimed
US-6495154-B1 ADMINISTERING ANTIDEPRESSANTS, ADRENERGIC STIMULANTS, SEROTONIN AGONISTS AND ANTAGONISTS AS THERAPEUTIC AGENTS FOR SEXUAL DISORDERS VIVUS INC. 2002-12-17 US claimed
EP-0126684-B1 DRUG DELIVERY SYSTEM UTILIZING THERMOSETTING GELS MERCK & CO. INC. (US) 1991-08-28 EP claimed
EP-0046270-B1 NOVEL DERIVATIVES OF BIO-AFFECTING PHENOLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITION CONTAINING THEM INTERx RESEARCH CORPORATION (US) 1986-05-21 EP claimed
EP-0152379-A2 Process for preparing pharmaceutical compositions containing unilamellar liposomes CIBA-GEIGY AG (CH) 1985-08-21 EP claimed