SCHEMBL2667937

SCHEMBL2667937

COc1cc(C(=O)Nc2ccc(C(=O)O)cn2)cc(S(=O)(=O)C(C)C)n1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GCK P35557 19/20 0.52
RARG P13631 2/20 0.49
RARA P10276 2/20 0.49
RARB P10826 2/20 0.49
HCAR3 P49019 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2656899 0.84 GCK (0.62) GCKRARGRARARARBHCAR3
SCHEMBL2667936 0.80 GCK (0.51) GCKRARGRARARARBHCAR3
SCHEMBL9070823 0.79 GCK (0.54) GCKRARGRARARARBHCAR3
SCHEMBL9070896 0.77 HCAR3 (0.52) GCKRARGRARARARBHCAR3
SCHEMBL2667682 0.77 GCK (0.59) GCKRARGRARARARBHCAR3
SCHEMBL2667765 0.76 GCK (0.65) GCKRARGRARARARB
SCHEMBL2657252 0.76 GCK (0.53) GCKRARGRARARARB
SCHEMBL2667952 0.76 GCK (0.57) GCKRARGRARARARB
SCHEMBL2667745 0.75 GCK (0.61) GCKRARGRARARARB
SCHEMBL9070871 0.74 GCK (0.66) GCKRARGRARARARBHCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009083553-A1 AZINE COMPOUNDS AS GLUCOKINASE ACTIVATORS RHEOSCIENCE A/S (DK) 2009-07-09 WO disclosed