SCHEMBL2668280

SCHEMBL2668280

CCCc1cc(OCc2cccnc2)cc(-c2nc3ncccc3[nH]2)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 3/20 0.54
AURKA O14965 4/20 0.48
FGFR1 P11362 1/20 0.46
FGFR2 P21802 1/20 0.46
FGFR3 P22607 1/20 0.46
DHODH Q02127 1/20 0.44
PDE5A O76074 5/20 0.44
PDE4A P27815 4/20 0.44
PDE4B Q07343 4/20 0.44
PDE4C Q08493 4/20 0.44
PDE4D Q08499 4/20 0.44
GRM2 Q14416 1/20 0.41
WNT1 P04628 2/20 0.41
NPY5R Q15761 1/20 0.40
MAOA P21397 1/20 0.40
DYRK1A Q13627 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL711302 0.89 PRMT5 (0.57) PRMT5AURKAFGFR1FGFR2FGFR3
SCHEMBL711172 0.78 PRMT5 (0.60) PRMT5AURKAFGFR1FGFR2FGFR3
SCHEMBL2668291 0.78 PRMT5 (0.65) PRMT5AURKADHODHPDE5APDE4A
SCHEMBL711966 0.72 PRMT5 (0.67) PRMT5AURKADHODHPDE5APDE4A
SCHEMBL711173 0.72 AURKA (0.56) PRMT5AURKAPDE5APDE4APDE4B
SCHEMBL2668141 0.72 DHODH (0.41) PRMT5DHODHGRM2MAOADYRK1A
SCHEMBL711692 0.71 PRMT5 (0.56) PRMT5AURKAFGFR1FGFR2FGFR3
SCHEMBL15972282 0.71 PRMT5 (1.00) PRMT5AURKADHODHPDE5APDE4A
SCHEMBL13639545 0.71 GRM5 (0.52) PRMT5FGFR1DHODHGRM2MAOA
SCHEMBL10206642 0.70 MAPK1 (0.47) PRMT5DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007028135-A2 IMIDAZOPYRIDINE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed