SCHEMBL26697211

SCHEMBL26697211

O=C(Nc1ccc(Br)cc1F)Nc1ccc(O)cc1Cl

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 6/20 0.65
LMNA P02545 5/20 0.65
KMT2A Q03164 4/20 0.65
MEN1 O00255 3/20 0.65
MAPT P10636 3/20 0.65
NPC1 O15118 3/20 0.59
RAB9A P51151 3/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
ALDH1A1 P00352 2/20 0.59
GAA P10253 1/20 0.54
HPGD P15428 1/20 0.54
ALOX12 P18054 1/20 0.54
CASP3 P42574 1/20 0.54
SENP7 Q9BQF6 1/20 0.54
SENP6 Q9GZR1 1/20 0.54
MAPK1 P28482 2/20 0.52
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA9 Q16790 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26697287 0.82 RAB9A (0.65) HTTLMNAKMT2AMEN1MAPT
SCHEMBL21750906 0.77 RAB9A (0.56) HTTKMT2AMEN1NPC1RAB9A
SCHEMBL29757932 0.77 RAB9A (0.56) HTTKMT2AMEN1NPC1RAB9A
SCHEMBL26697245 0.76 RAB9A (0.53) HTTLMNAKMT2AMEN1MAPT
SCHEMBL17161297 0.75 LMNA (0.65) HTTLMNAKMT2AMEN1MAPT
SCHEMBL20560335 0.75 NPC1 (0.59) HTTLMNAKMT2AMEN1MAPT
SCHEMBL21834398 0.75 NPC1 (1.00) HTTLMNAKMT2AMEN1MAPT
SCHEMBL28460880 0.74 MAPT (0.49) HTTLMNAKMT2AMEN1MAPT
SCHEMBL27915487 0.74 LMNA (0.59) HTTLMNAKMT2AMEN1MAPT
SCHEMBL21750964 0.74 KDR (0.57) KMT2AMEN1MAPTGAACA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114920703-B Quinazoline derivative and preparation method and application thereof 天津济坤医药科技有限公司 2024-01-09 CN disclosed
WO-2023226323-A1 QUINAZOLINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 天津济坤医药科技有限公司 2023-11-30 WO disclosed
WO-2023226323-A1 QUINAZOLINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 天津济坤医药科技有限公司 2023-11-30 WO disclosed
CN-114920703-A Quinazoline derivative and preparation method and application thereof 天津济坤医药科技有限公司 2022-08-19 CN disclosed